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Ureidopyridazine derivatives as Acyl-CoA:cholesterol acyltransferase inhibitors 1-gen-2006 Gelain, Arianna; Bettinelli, Ilaria; Barlocco, Daniela; KWON Byoung, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio
3-Heptylamino-5-phenylpyridazine derivatives as analogues of acyl-CoA: cholesterol acyltransferase inhibitors containing the N-heptyl-N’-arylureidic moiety 1-gen-2006 Gelain, Arianna; Barlocco, Daniela; KWON Byong, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio
Alternative mechanistic paths in the hetero-Diels-Alder reaction of alpha-oxothiones: a theoretical study 1-gen-2007 Legnani, Laura; Lunghi, Carlotta; Marinone, Franca; Nativi, Cristina; Richichi, Barbara; Toma, Lucio
A full conformational characterization of 13-ethylprogestogens through theoretical calculations and nuclear magnetic resonance spectroscopy 1-gen-2007 Colombo, Diego; Ferraboschi, Patrizia; Legnani, Laura; Prestileo, Paolo; Toma, Lucio
Synthesis, conformational studies, binding assessment and liposome insertion of a thioether-bridged mimetic of the antigen GM3 ganglioside lactone 1-gen-2007 Toma, Lucio; Di Cola, Emanuela; Ienco, Andrea; Legnani, Laura; Lunghi, Carlotta; Moneti, Gloriano; Richichi, Barbara; Ristori, Sandra; Dell'Atti, Daniela; Nativi, Cristina
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors 1-gen-2008 Murineddu, Gabriele; Murruzzu, Caterina; Curzu Maria, M; Chelucci, Giorgio; Gotti, Cecilia; Gaimarri, Annalisa; Legnani, Laura; Toma, Lucio; Pinna Gerard, A.
Biphenyl versus Phenylpyridazine Derivatives: The Role of the Heterocycle in a Series of Acyl-CoA:Cholesterol Acyl Transferase Inhibitors 1-gen-2008 Gelain, Arianna; Barlocco, Daniela; Kwon Byoung, Mog; Jeong Tae, Sook; Im Kyung, Ran; Legnani, Laura; Toma, Lucio
Complete 1H and 13C assignments of (21R) and (21S) diastereomers of argatroban 1-gen-2008 Colombo, Diego; Ferraboschi, Patrizia; Grisenti, Paride; Legnani, Laura
A new stereoselective approach to a selectively protected derivative of D-pinitol and its evaluation as alpha-L-rhamnopyranose mimetic 1-gen-2008 Catelani, Giorgio; D'Andrea, Felicia; Griselli, Alessio; Guazzelli, Lorenzo; Legnani, Laura; Toma, Lucio
A full conformational characterization of natural ionones and irones, as well as 13-alkyl-substituted alpha-ionones 1-gen-2008 Legnani, Laura; Luparia, Marco; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni
Enantioselective Synthesis and Olfactory Evaluation of Bicyclic r- andγ-Ionone Derivatives: The 3D Arrangement of Key Molecular FeaturesRelevant to the Violet Odor of Ionones 1-gen-2009 Luparia, Marco; Legnani, Laura; Porta, Alessio; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni
Cyclic glycopeptidomimetics through a versatile sugar-based scaffold 1-gen-2009 Altamura, Maria; Dragoni, Elisa; Infantino Angela, Simona; Legnani, Laura; Ludbrook Steve, B.; Menchi, Gloria; Toma, Lucio; Nativi, Cristina
An exhaustive conformational evaluation of the HIV-1 inhibitor BMS-378806 through theoretical calculations and nuclear magnetic resonance spectroscopy 1-gen-2009 Colombo, Diego; Villa, Stefania; Solano, Lucrezia; Legnani, Laura; Marinone, Franca; Toma, Lucio
Modeling of synthetic phosphono and carba analogues ofN-acetyl-alpha-D-mannosamine 1-phosphate, the repeating unit of the capsular polysaccharide from Neisseria meningitidis serovar A 1-gen-2009 Toma, Lucio; Legnani, Laura; Rencurosi, Anna; Poletti, Laura; Lay, Luigi; Russo, Giovanni
Synthesis, molecular dynamics simulations, and biology of a carba-analogue of the trisaccharide repeating unit of Streptococcus pneumoniae 19F capsular polysaccharide 1-gen-2009 Legnani, Laura; Ronchi, Silvia; Fallarini, Silvia; Lombardi, Grazia; Campo, Federica; Panza, Luigi; Lay, Luigi; Poletti, Laura; Toma, Lucio; Ronchetti, Fiamma; Compostella, Federica
Stable GM3 Lactone Mimetic Raises Antibodies Specific for the Antigens Expressed on Melanoma Cells 1-gen-2010 Arcangeli, Annarosa; Toma, Lucio; Contiero, Luca; Crociani, Olivia; Legnani, Laura; Lunghi, Carlotta; Nesti, Elisa; Moneti, Gloriano; Richichi, Barbara; Nativi, Cristina
Synthesis, modeling, and crystallographic study of 3,4-disubstituted-1,2,5-oxadiazoles and evaluation of their ability to decrease STAT3 activity 1-gen-2010 Shin Dae, Seop; Masciocchi, Daniela; Gelain, Arianna; Villa, Stefania; Barlocco, Daniela; Meneghetti, Fiorella; Pedretti, Alessandro; Han Young, Min; Han Dong, Cho; Kwon Byoung, Mog; Legnani, Laura; Toma, Lucio
Modeling and Spectroscopic Studies of Synthetic Diazabicyclo Analogs of the HIV-1 Inhibitor BMS-378806 and Evaluation of Their Antiviral Activity 1-gen-2011 Legnani, Laura; Colombo, Diego; Cocchi, Elena; Solano, Lucrezia; Villa, Stefania; Lopalco, Lucia; Asti, Valeria; Diomede, Lorenzo; Marinone, Franca; Toma, Lucio
Molecular dynamics simulations of the Salmonella typhi Vi antigenic polysaccharide and effects of the introduction of a zwitterionic motif 1-gen-2011 Legnani, Laura; Compostella, Federica; Grazioso, Giovanni; Marinone, Franca; Toma, Lucio
Mechanism of falcipain-2 inhibition by a,b-unsaturated benzo[1,4]diazepin-2-one methyl ester 1-gen-2012 Grazioso, G.; Legnani, Laura; Toma, Lucio; Ettari, R.; Micale, N.; De Micheli, C.
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