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Functional investigation of the antitubercular drug target Decaprenylphosphoryl-β-D-ribofuranose-2-epimerase DprE1/DprE2 complex 1-gen-2022 Sammartino, Josè Camilla; Morici, Martino; Stelitano, Giovanni; Degiacomi, Giulia; Riccardi, Giovanna; Chiarelli, Laurent Roberto
Synthesis and assessment of the in vitro and ex vivo activity of salicylate synthase (Mbti) inhibitors as new candidates for the treatment of mycobacterial infections 1-gen-2022 Mori, M; Stelitano, G; Griego, A; Chiarelli, Lr; Cazzaniga, G; Gelain, A; Pini, E; Camera, M; Canzano, P; Fumagalli, A; Scarpa, E; Cordiglieri, C; Rizzello, L; Villa, S; Meneghetti, F.
Characterization of mycobacterial enzymes as targets for potential antitubercular compounds. 4-apr-2022 Stelitano, Giovanni
CanB, a Druggable Cellular Target in Mycobacterium tuberculosis 1-gen-2023 Degiacomi, Giulia; Gianibbi, Beatrice; Recchia, Deborah; Stelitano, Giovanni; Truglio, Giuseppina Ivana; Marra, Paola; Stamilla, Alessandro; Makarov, Vadim; Chiarelli, Laurent Robert; Manetti, Fabrizio; Pasca, Maria Rosalia
Mycobacterium abscessus Infections in Cystic Fibrosis Individuals: A Review on Therapeutic Options 1-gen-2023 Recchia, Deborah; Stelitano, Giovanni; Stamilla, Alessandro; Gutierrez, Damaris L; Degiacomi, Giulia; Chiarelli, Laurent R; Pasca, Maria Rosalia
Mycobacterium abscessus siderophores biosynthesis as a target to inhibit the iron uptake mechanism 1-gen-2023 Cocorullo, Mario; Stelitano, Giovanni; Mori, Matteo; Cazzaniga, Giulia; Roversi, Martina; Covaceuszach, Sonia; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, Laurent R.
From virulence factors to drug development: MbtI as an effective Mycobacterium tuberculosis target 1-gen-2023 Stelitano, Giovanni; Cocorullo, Mario; Cazzaniga, Giulia; Mori, Matteo; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, LAURENT ROBERT
Moles of Molecules against Mycobacterium abscessus: A Review of Current Research 1-gen-2023 Cocorullo, Mario; Bettoni, Christian; Foiadelli, Sara; Stelitano, Giovanni
Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity 1-gen-2023 Dongguang, F; Wang, B; Stelitano, G; Savková, K; Riabova, O; Shi, R; Wu, X; Chiarelli, Lr; Mikušová, K; Makarov, V; Lu, Y; Hong, H; Qiao, C.
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? 1-gen-2023 D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona
Improve protection to prevent infections: application of reverse vaccinology against cystic fibrosis pathogens. 1-gen-2023 Cocorullo, M; Chiarelli, Lr; Stelitano, G
Targeting Siderophore-Mediated Iron Uptake in M. abscessus: A New Strategy to Limit the Virulence of Non-Tuberculous Mycobacteria. 1-gen-2023 Mori, M; Stelitano, G; Cazzaniga, G; Gelain, A; Tresoldi, A; Cocorullo, M; Roversi, M; Chiarelli, Lr; Tomaiuolo, M; Del Re, P; Mangiatordi, Gf; Griego, A; Rizzello, L; Cassetta, A; Covaceuszach, S; Villa, S; Meneghetti, F.
Iron Acquisition and Metabolism as a Promising Target for Antimicrobials (Bottlenecks and Opportunities): Where Do We Stand? 1-gen-2023 Stelitano, Giovanni; Cocorullo, Mario; Mori, Matteo; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, LAURENT ROBERT
Structural basis for specific inhibition of salicylate synthase from Mycobacterium abscessus 1-gen-2024 Mori, M; Cocorullo, M; Tresoldi, A; Cazzaniga, G; Gelain, A; Stelitano, G; Chiarelli, Lr; Tomaiuolo, M; Del Re, P; Mangiatordi, Gf; Garofalo, M; Cassetta, A; Covaceuszach, S; Villa, S; Meneghetti, F.
Benzothiozinone derivatives with anti-tubercular Activity−Further side chain investigation 1-gen-2024 Wu, X.; Wang, W.; Stelitano, G.; Riabova, O.; Wang, B.; Niu, W.; Cocorullo, M.; Shi, R.; Chiarelli, L. R.; Makarov, V.; Lu, Y.; Li, C.; Qiao, C.
Mostrati risultati da 21 a 35 di 35
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