STELITANO, GIOVANNI

STELITANO, GIOVANNI  

DIPARTIMENTO DI BIOLOGIA E BIOTECNOLOGIE "LAZZARO SPALLANZANI"  

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Risultati 1 - 20 di 35 (tempo di esecuzione: 0.017 secondi).
Titolo Data di pubblicazione Autore(i) File
A dual-target approach in anti-tuberculosis therapy: new MptpB/MbtI. 1-gen-2020 Cazzaniga, G; Mori, M; Gelain, A; Pini, E; Stelitano, G; Chiarelli, Lr; Meneghetti, F; Villa, S.
A multitarget approach to drug discovery inhibiting Mycobacterium tuberculosis MbtI and MPtpB 1-gen-2021 Stelitano, G; Cazzaniga, G; Mori, M; Villa, S; Meneghetti, F; Chiarelli, Lr.
Benzothiozinone derivatives with anti-tubercular Activity−Further side chain investigation 1-gen-2024 Wu, X.; Wang, W.; Stelitano, G.; Riabova, O.; Wang, B.; Niu, W.; Cocorullo, M.; Shi, R.; Chiarelli, L. R.; Makarov, V.; Lu, Y.; Li, C.; Qiao, C.
CanB, a Druggable Cellular Target in Mycobacterium tuberculosis 1-gen-2023 Degiacomi, Giulia; Gianibbi, Beatrice; Recchia, Deborah; Stelitano, Giovanni; Truglio, Giuseppina Ivana; Marra, Paola; Stamilla, Alessandro; Makarov, Vadim; Chiarelli, Laurent Robert; Manetti, Fabrizio; Pasca, Maria Rosalia
Characterization of mycobacterial enzymes as targets for potential antitubercular compounds. 4-apr-2022 Stelitano, Giovanni
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? 1-gen-2023 D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona
Development of 6-Methanesulfonyl-8-nitrobenzothiazinone Based Antitubercular Agents 1-gen-2022 Shi, R.; Wang, B.; Stelitano, G.; Wu, X.; Shan, Y.; Wu, Y.; Wang, X.; Chiarelli, L. R.; Lu, Y.; Qiao, C.
Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents 1-gen-2018 Chiarelli, Laurent R; Mori, Matteo; Barlocco, Daniela; Beretta, Giangiacomo; Gelain, Arianna; Pini, Elena; Porcino, Marianna; Mori, Giorgia; Stelitano, Giovanni; Costantino, Luca; Lapillo, Margherita; Bonanni, Davide; Poli, Giulio; Tuccinardi, Tiziano; Villa, Stefania; Meneghetti, Fiorella
Exploring the role of the heterocyclic moiety of 5-(4-nitrophenyl)-2-furoic acid, a promising inhibitor of MbtI from Mycobacterium tuberculosis. 1-gen-2019 Mori, M; Chiarelli, Lr; Stelitano, G; Gelain, A; Tuccinardi, T; Bellinzoni, M.; Meneghetti, F; Villa, S.
From virulence factors to drug development: MbtI as an effective Mycobacterium tuberculosis target 1-gen-2023 Stelitano, Giovanni; Cocorullo, Mario; Cazzaniga, Giulia; Mori, Matteo; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, LAURENT ROBERT
Functional investigation of the antitubercular drug target Decaprenylphosphoryl-β-D-ribofuranose-2-epimerase DprE1/DprE2 complex 1-gen-2022 Sammartino, Josè Camilla; Morici, Martino; Stelitano, Giovanni; Degiacomi, Giulia; Riccardi, Giovanna; Chiarelli, Laurent Roberto
Improve protection to prevent infections: application of reverse vaccinology against cystic fibrosis pathogens. 1-gen-2023 Cocorullo, M; Chiarelli, Lr; Stelitano, G
Investigating the inhibition mechanism and catalytic cycle of MbtI, the salicylate synthase from Mycobacterium tuberculosis. 1-gen-2020 Mori, M.; Villa, S.; Gelain, A; Pini, E. R. E.; Stelitano, G.; Chiarelli, L. R.; Tuccinardi, T.; Bellinzoni, M.; Meneghetti, F.
Iron Acquisition and Metabolism as a Promising Target for Antimicrobials (Bottlenecks and Opportunities): Where Do We Stand? 1-gen-2023 Stelitano, Giovanni; Cocorullo, Mario; Mori, Matteo; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, LAURENT ROBERT
Moles of Molecules against Mycobacterium abscessus: A Review of Current Research 1-gen-2023 Cocorullo, Mario; Bettoni, Christian; Foiadelli, Sara; Stelitano, Giovanni
Multi-target antitubercular drugs: identification of novel dual MbtI and MptpB inhibitors. 1-gen-2019 Mori, M; Villa, S; Chiarelli, Lr; Stelitano, G; Gelain, A; Tuccinardi, T; Bellinzoni, M.; Meneghetti, F.
Multitargeting Compounds: A Promising Strategy to Overcome Multi-Drug Resistant Tuberculosis 1-gen-2020 Stelitano, Giovanni; Sammartino, José Camilla; Chiarelli, Laurent Roberto
Mycobacterium abscessus Infections in Cystic Fibrosis Individuals: A Review on Therapeutic Options 1-gen-2023 Recchia, Deborah; Stelitano, Giovanni; Stamilla, Alessandro; Gutierrez, Damaris L; Degiacomi, Giulia; Chiarelli, Laurent R; Pasca, Maria Rosalia
Mycobacterium abscessus siderophores biosynthesis as a target to inhibit the iron uptake mechanism 1-gen-2023 Cocorullo, Mario; Stelitano, Giovanni; Mori, Matteo; Cazzaniga, Giulia; Roversi, Martina; Covaceuszach, Sonia; Villa, Stefania; Meneghetti, Fiorella; Chiarelli, Laurent R.
New insight into structure-activity of furan-based salicylate synthase (MbtI) inhibitors as potential antitubercular agents 1-gen-2019 Chiarelli, Laurent R; Mori, Matteo; Beretta, Giangiacomo; Gelain, Arianna; Pini, Elena; Sammartino, Josè Camilla; Stelitano, Giovanni; Barlocco, Daniela; Costantino, Luca; Lapillo, Margherita; Poli, Giulio; Caligiuri, Isabella; Rizzolio, Flavio; Bellinzoni, Marco; Tuccinardi, Tiziano; Villa, Stefania; Meneghetti, Fiorella