Sfoglia per Rivista ACS INFECTIOUS DISEASES
A Coumarin-Based Analogue of Thiacetazone as Dual Covalent Inhibitor and Potential Fluorescent Label of HadA in Mycobacterium tuberculosis
2021-01-01 Farjallah, Asma; Chiarelli, Laurent R; Forbak, Martin; Degiacomi, Giulia; Danel, Mathieu; Goncalves, Fernanda; Carayon, Chantal; Seguin, Cendrine; Fumagalli, Marco; Záhorszká, Monika; Vega, Elodie; Abid, Souhir; Grzegorzewicz, Anna; Jackson, Mary; Peixoto, Antonio; Korduláková, Jana; Pasca, Maria Rosalia; Lherbet, Christian; Chassaing, Stefan
Design and Synthesis of Pyrano[3,2-b]indolones Showing Antimycobacterial Activity
2021-01-01 Monakhova, N.; Kordulakova, J.; Vocat, A.; Egorova, A.; Lepioshkin, A.; Salina, E. G.; Nosek, J.; Repkova, E.; Zemanova, J.; Jurdakova, H.; Gorova, R.; Roh, J.; Degiacomi, G.; Sammartino, J. C.; Pasca, M. R.; Cole, S. T.; Mikusova, K.; Makarov, V.
Design, Synthesis, and Antiviral Evaluation of Sialic Acid Derivatives as Inhibitors of Newcastle Disease Virus Hemagglutinin-Neuraminidase: A Translational Study on Human Parainfluenza Viruses
2023-01-01 Rota, Paola; La Rocca, Paolo; Bonfante, Francesco; Pagliari, Matteo; Piccoli, Marco; Cirillo, Federica; Ghiroldi, Andrea; Franco, Valentina; Pappone, Carlo; Allevi, Pietro; Anastasia, Luigi
Designing Probes for Immunodiagnostics: Structural Insights into an Epitope Targeting Burkholderia Infections
2017-01-01 Capelli, Riccardo; Matterazzo, Elena; Arnabili, Marco; Peri, Claudio; Gori, Alessandro; Gagni, Paola; Chiari, Marcella; Lertmemongkolchai, Ganjana; Cretich, Marina; Bolognesi, Martino; Colombo, Giorgio; Gourlay, Louise J.
Enhancing Antibody Serodiagnosis Using a Controlled Peptide Coimmobilization Strategy
2018-01-01 Sola, Laura; Gagni, Paola; D'Annessa, Ilda; Capelli, Riccardo; Bertino, Camilla; Romanato, Alessandro; Damin, Francesco; Bergamaschi, Greta; Marchisio, Edoardo; Cuzzocrea, Angela; Bombaci, Mauro; Grifantini, Renata; Chiari, Marcella; Colombo, Giorgio; Gori, Alessandro; Cretich, Marina
Flexible vs Rigid Epitope Conformations for Diagnostic- and Vaccine-Oriented Applications: Novel Insights from the Burkholderia pseudomallei BPSL2765 Pa13 Epitope
2016-01-01 Gori, Alessandro; Peri, Claudio; Quilici, Giacomo; Nithichanon, Arnone; Gaudesi, Davide; Longhi, Renato; Gourlay Louise, J; Bolognesi, Martino; Lertmemongkolchai, Ganjana; Musco, Giovanna; Colombo, Giorgio
GM-3 Lactone Mimetic Interacts with CD4 and HIV-1 Env Proteins, Hampering HIV-1 Infection without Inducing a Histopathological Alteration
2016-01-01 Richichi, Barbara; Pastori, Claudia; Gherardi, Stefano; Venuti, Assunta; Cerreto, Antonella; Sanvito, Francesca; Toma, Lucio; Lopalco, Lucia; Nativi, Cristina
Naphthalene Diimide–Tetraazacycloalkane Conjugates Are G-Quadruplex-Based HIV-1 Inhibitors with a Dual Mode of Action
2024-01-01 Nadai, Matteo; Doria, Filippo; Frasson, Ilaria; Perrone, Rosalba; Pirota, Valentina; Bergamaschi, Greta; Freccero, Mauro; Richter, Sara N.
New insights into the mechanism of action of the thienopyrimidine antitubercular prodrug TP053
2020-01-01 Chiarelli, Lr; Salina, Eg; Mori, G; Azhikina, T; Riabova, O; Lepioshkin, A; Grigorov, A; Forbak, M; Madacki, J; Orena, Bs; Manfredi, M; Gosetti, F; Buzzi, A; Degiacomi, G; Sammartino, Jc; Marengo, E; Korduláková, J; Riccardi, G; Mikušová, K; Makarov, V; Pasca, Mr.
A phenotypic based target screening approach delivers new antitubercular CTP synthetase inhibitors
2017-01-01 Esposito, Marta; Szadocka, Sára; Degiacomi, Giulia; Orena, BEATRICE SILVIA; Mori, Giorgia; Piano, Valentina; Boldrin, Francesca; Zemanova, Julia; Huszár, Stanislav; Barros, David; Ekins, Sean; Lelièvre, Joël; Manganelli, Riccardo; Mattevi, Andrea; Pasca, MARIA ROSALIA; Riccardi, Giovanna; Ballell, Lluis; Mikušová, Katarína; Chiarelli, Laurent
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors
2019-01-01 Landi, G.; Linciano, P.; Borsari, C.; Bertolacini, C. P.; Moraes, C. B.; Cordeiro-Da-Silva, A.; Gul, S.; Witt, G.; Kuzikov, M.; Costi, M. P.; Pozzi, C.; Mangani, S.
Ten Years with New Delhi Metallo-β-lactamase-1 (NDM-1): From Structural Insights to Inhibitor Design
2019-01-01 Linciano, P.; Cendron, L.; Gianquinto, E.; Spyrakis, F.; Tondi, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A Coumarin-Based Analogue of Thiacetazone as Dual Covalent Inhibitor and Potential Fluorescent Label of HadA in Mycobacterium tuberculosis | 1-gen-2021 | Farjallah, Asma; Chiarelli, Laurent R; Forbak, Martin; Degiacomi, Giulia; Danel, Mathieu; Goncalves, Fernanda; Carayon, Chantal; Seguin, Cendrine; Fumagalli, Marco; Záhorszká, Monika; Vega, Elodie; Abid, Souhir; Grzegorzewicz, Anna; Jackson, Mary; Peixoto, Antonio; Korduláková, Jana; Pasca, Maria Rosalia; Lherbet, Christian; Chassaing, Stefan | |
Design and Synthesis of Pyrano[3,2-b]indolones Showing Antimycobacterial Activity | 1-gen-2021 | Monakhova, N.; Kordulakova, J.; Vocat, A.; Egorova, A.; Lepioshkin, A.; Salina, E. G.; Nosek, J.; Repkova, E.; Zemanova, J.; Jurdakova, H.; Gorova, R.; Roh, J.; Degiacomi, G.; Sammartino, J. C.; Pasca, M. R.; Cole, S. T.; Mikusova, K.; Makarov, V. | |
Design, Synthesis, and Antiviral Evaluation of Sialic Acid Derivatives as Inhibitors of Newcastle Disease Virus Hemagglutinin-Neuraminidase: A Translational Study on Human Parainfluenza Viruses | 1-gen-2023 | Rota, Paola; La Rocca, Paolo; Bonfante, Francesco; Pagliari, Matteo; Piccoli, Marco; Cirillo, Federica; Ghiroldi, Andrea; Franco, Valentina; Pappone, Carlo; Allevi, Pietro; Anastasia, Luigi | |
Designing Probes for Immunodiagnostics: Structural Insights into an Epitope Targeting Burkholderia Infections | 1-gen-2017 | Capelli, Riccardo; Matterazzo, Elena; Arnabili, Marco; Peri, Claudio; Gori, Alessandro; Gagni, Paola; Chiari, Marcella; Lertmemongkolchai, Ganjana; Cretich, Marina; Bolognesi, Martino; Colombo, Giorgio; Gourlay, Louise J. | |
Enhancing Antibody Serodiagnosis Using a Controlled Peptide Coimmobilization Strategy | 1-gen-2018 | Sola, Laura; Gagni, Paola; D'Annessa, Ilda; Capelli, Riccardo; Bertino, Camilla; Romanato, Alessandro; Damin, Francesco; Bergamaschi, Greta; Marchisio, Edoardo; Cuzzocrea, Angela; Bombaci, Mauro; Grifantini, Renata; Chiari, Marcella; Colombo, Giorgio; Gori, Alessandro; Cretich, Marina | |
Flexible vs Rigid Epitope Conformations for Diagnostic- and Vaccine-Oriented Applications: Novel Insights from the Burkholderia pseudomallei BPSL2765 Pa13 Epitope | 1-gen-2016 | Gori, Alessandro; Peri, Claudio; Quilici, Giacomo; Nithichanon, Arnone; Gaudesi, Davide; Longhi, Renato; Gourlay Louise, J; Bolognesi, Martino; Lertmemongkolchai, Ganjana; Musco, Giovanna; Colombo, Giorgio | |
GM-3 Lactone Mimetic Interacts with CD4 and HIV-1 Env Proteins, Hampering HIV-1 Infection without Inducing a Histopathological Alteration | 1-gen-2016 | Richichi, Barbara; Pastori, Claudia; Gherardi, Stefano; Venuti, Assunta; Cerreto, Antonella; Sanvito, Francesca; Toma, Lucio; Lopalco, Lucia; Nativi, Cristina | |
Naphthalene Diimide–Tetraazacycloalkane Conjugates Are G-Quadruplex-Based HIV-1 Inhibitors with a Dual Mode of Action | 1-gen-2024 | Nadai, Matteo; Doria, Filippo; Frasson, Ilaria; Perrone, Rosalba; Pirota, Valentina; Bergamaschi, Greta; Freccero, Mauro; Richter, Sara N. | |
New insights into the mechanism of action of the thienopyrimidine antitubercular prodrug TP053 | 1-gen-2020 | Chiarelli, Lr; Salina, Eg; Mori, G; Azhikina, T; Riabova, O; Lepioshkin, A; Grigorov, A; Forbak, M; Madacki, J; Orena, Bs; Manfredi, M; Gosetti, F; Buzzi, A; Degiacomi, G; Sammartino, Jc; Marengo, E; Korduláková, J; Riccardi, G; Mikušová, K; Makarov, V; Pasca, Mr. | |
A phenotypic based target screening approach delivers new antitubercular CTP synthetase inhibitors | 1-gen-2017 | Esposito, Marta; Szadocka, Sára; Degiacomi, Giulia; Orena, BEATRICE SILVIA; Mori, Giorgia; Piano, Valentina; Boldrin, Francesca; Zemanova, Julia; Huszár, Stanislav; Barros, David; Ekins, Sean; Lelièvre, Joël; Manganelli, Riccardo; Mattevi, Andrea; Pasca, MARIA ROSALIA; Riccardi, Giovanna; Ballell, Lluis; Mikušová, Katarína; Chiarelli, Laurent | |
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors | 1-gen-2019 | Landi, G.; Linciano, P.; Borsari, C.; Bertolacini, C. P.; Moraes, C. B.; Cordeiro-Da-Silva, A.; Gul, S.; Witt, G.; Kuzikov, M.; Costi, M. P.; Pozzi, C.; Mangani, S. | |
Ten Years with New Delhi Metallo-β-lactamase-1 (NDM-1): From Structural Insights to Inhibitor Design | 1-gen-2019 | Linciano, P.; Cendron, L.; Gianquinto, E.; Spyrakis, F.; Tondi, D. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile