Sfoglia per Autore
Small molecule integrin antagonists in cancer therapy
2009-01-01 Paolillo, Mayra; Russo, MARIKA ALESSANDRA; Serra, Massimo; Colombo, Lino; Schinelli, Sergio
Novel stereoselective syntheses of (2E,4E)-4-(4,4-dimethylpent-2-ynylidene)-N1,N5-dimethyl-N1,N5-bis(naphthalen-1-ylmethyl)pent-2-ene-1,5-diamine
2009-01-01 Colombo, Lino; DI GIACOMO, Marcello; Serra, Massimo; Tambini, SIMONE MARIA
Process for the preparation of keto intermediates
2010-01-01 Attolino, Emanuele; Colombo, Lino; Zurlo Ada, Maria; Artico, Marco; Allegrini, Pietro
Process for the production of sitagliptin
2010-01-01 Rasparini, Marcello; Colombo, Lino; D'Arienzo, Giuseppe; Tufaro, Roberto; Venegoni, Serena
Method for the preparation of Rufinamide
2010-01-01 Attolino, Emanuele; Colombo, Lino; Mormino, Ilaria; Allegrini, Pietro
Stereoselective Pd-catalyzed synthesis of quaternary a-C-D-mannosyl-(S)-amino acids
2011-01-01 DI GIACOMO, Marcello; Serra, Massimo; Brusasca, Marco; Colombo, Lino
Effect of tetracyclines on the dynamics of formation and destructuration of {beta}2-microglobulin amyloid fibrils.
2011-01-01 Giorgetti, Sofia; Raimondi, Sara; Pagano, K; Relini, A; Bucciantini, M; Corazza, A; Fogolari, F; Codutti, L; Salmona, M; Mangione, Palma; Colombo, Lino; De Luigi, A; Porcari, Riccardo; Gliozzi, A; Stefani, M; Esposito, G; Bellotti, Vittorio; Stoppini, Monica
A small-molecule RGD-integrin antagonist inhibits cell adhesion, cell migration and induces anoikis in glioblastoma cells.
2013-01-01 Russo, Ma; Paolillo, Mayra; Sanchez Hernandez, Y; Curti, Daniela; Ciusani, E; Serra, Massimo; Colombo, Lino; Schinelli, Sergio
In-Solution Structural Considerations by1H NMR and Solid-State Thermal Properties of Inulin-d-α-Tocopherol Succinate (INVITE) Micelles as Drug Delivery Systems for Hydrophobic Drugs
2014-01-01 Catenacci, Laura; Delia, Mandracchia; Sorrenti, MILENA LILLINA; Colombo, Lino; Serra, Massimo; Tripodo, Giuseppe
Synthesis of Easy-to-Functionalize Azabicycloalkane Scaffolds as Dipeptide Turn Mimics en Route to cRGD-Based Bioconjugates
2015-01-01 Serra, Massimo; Tambini, SIMONE MARIA; DI GIACOMO, Marcello; Peviani, ELENA GIULIA; Belvisi, Laura; Colombo, Lino
Synthesis of Variously Functionalized Azabicycloalkane Scaffolds by Domino Metathesis Reactions
2017-01-01 Serra, Massimo; Peviani, Elena Giulia; Bernardi, Eric; Colombo, Lino
One-Pot Vinylation of Azlactones: Fast Access to Enantioenriched α-Vinyl Quaternary Amino Acids
2017-01-01 Serra, Massimo; Bernardi, Eric; Marrubini, Giorgio; Colombo, Lino
Synthesis of differently bioconjugated novel c-RGD antagonist
2018-01-01 Bernardi, Eric; Serra, Massimo; Protti, Stefano; Fagnoni, Maurizio; Perteghella, Sara; Bari, Elia; Colombo, Lino
An RGD small-molecule integrin antagonist induces detachment-mediated anoikis in glioma cancer stem cells
2018-01-01 Paolillo, Mayra; Galiazzo, Marisa C.; Daga, Antonio; Ciusani, Emilio; Serra, Massimo; Colombo, Lino; Schinelli, Sergio
Synthesis of functionalized 6,5- and 7,5-azabicycloalkane amino acids by metathesis reactions
2019-01-01 Serra, M.; Bernardi, E.; De Lorenzi, E.; Colombo, L.
Palladium-catalyzed asymmetric decarboxylative allylation of azlactone enol carbonates: Fast access to enantioenriched α-allyl quaternary amino acids
2019-01-01 Serra, M; Bernardi, E; Marrubini, G; De Lorenzi, E; Colombo, L
One-Pot Preparation of Functionalized Azabicyclo[6.3.0]alkanone Amino Acids by Tandem Cross Enyne Metathesis/Ring-Closing Metathesis
2020-01-01 Bernardi, E.; Colombo, L.; De Lorenzi, E.; Carraro, M.; Serra, M.
Recent Advances in One-Pot Enyne Metathesis Processes for the Preparation of Biologically and Medicinally Relevant Compounds
2021-01-01 Bernardi, E.; Colombo, L.; Serra, M.
Synthesis of Functionalized Proline-Derived Azabicycloalkane Amino Acids and Their Applications in Drug Discovery: Recent Advances
2023-01-01 Serra, M.; Terreni, M.; Bernardi, E.; Colombo, L.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Small molecule integrin antagonists in cancer therapy | 1-gen-2009 | Paolillo, Mayra; Russo, MARIKA ALESSANDRA; Serra, Massimo; Colombo, Lino; Schinelli, Sergio | |
Novel stereoselective syntheses of (2E,4E)-4-(4,4-dimethylpent-2-ynylidene)-N1,N5-dimethyl-N1,N5-bis(naphthalen-1-ylmethyl)pent-2-ene-1,5-diamine | 1-gen-2009 | Colombo, Lino; DI GIACOMO, Marcello; Serra, Massimo; Tambini, SIMONE MARIA | |
Process for the preparation of keto intermediates | 1-gen-2010 | Attolino, Emanuele; Colombo, Lino; Zurlo Ada, Maria; Artico, Marco; Allegrini, Pietro | |
Process for the production of sitagliptin | 1-gen-2010 | Rasparini, Marcello; Colombo, Lino; D'Arienzo, Giuseppe; Tufaro, Roberto; Venegoni, Serena | |
Method for the preparation of Rufinamide | 1-gen-2010 | Attolino, Emanuele; Colombo, Lino; Mormino, Ilaria; Allegrini, Pietro | |
Stereoselective Pd-catalyzed synthesis of quaternary a-C-D-mannosyl-(S)-amino acids | 1-gen-2011 | DI GIACOMO, Marcello; Serra, Massimo; Brusasca, Marco; Colombo, Lino | |
Effect of tetracyclines on the dynamics of formation and destructuration of {beta}2-microglobulin amyloid fibrils. | 1-gen-2011 | Giorgetti, Sofia; Raimondi, Sara; Pagano, K; Relini, A; Bucciantini, M; Corazza, A; Fogolari, F; Codutti, L; Salmona, M; Mangione, Palma; Colombo, Lino; De Luigi, A; Porcari, Riccardo; Gliozzi, A; Stefani, M; Esposito, G; Bellotti, Vittorio; Stoppini, Monica | |
A small-molecule RGD-integrin antagonist inhibits cell adhesion, cell migration and induces anoikis in glioblastoma cells. | 1-gen-2013 | Russo, Ma; Paolillo, Mayra; Sanchez Hernandez, Y; Curti, Daniela; Ciusani, E; Serra, Massimo; Colombo, Lino; Schinelli, Sergio | |
In-Solution Structural Considerations by1H NMR and Solid-State Thermal Properties of Inulin-d-α-Tocopherol Succinate (INVITE) Micelles as Drug Delivery Systems for Hydrophobic Drugs | 1-gen-2014 | Catenacci, Laura; Delia, Mandracchia; Sorrenti, MILENA LILLINA; Colombo, Lino; Serra, Massimo; Tripodo, Giuseppe | |
Synthesis of Easy-to-Functionalize Azabicycloalkane Scaffolds as Dipeptide Turn Mimics en Route to cRGD-Based Bioconjugates | 1-gen-2015 | Serra, Massimo; Tambini, SIMONE MARIA; DI GIACOMO, Marcello; Peviani, ELENA GIULIA; Belvisi, Laura; Colombo, Lino | |
Synthesis of Variously Functionalized Azabicycloalkane Scaffolds by Domino Metathesis Reactions | 1-gen-2017 | Serra, Massimo; Peviani, Elena Giulia; Bernardi, Eric; Colombo, Lino | |
One-Pot Vinylation of Azlactones: Fast Access to Enantioenriched α-Vinyl Quaternary Amino Acids | 1-gen-2017 | Serra, Massimo; Bernardi, Eric; Marrubini, Giorgio; Colombo, Lino | |
Synthesis of differently bioconjugated novel c-RGD antagonist | 1-gen-2018 | Bernardi, Eric; Serra, Massimo; Protti, Stefano; Fagnoni, Maurizio; Perteghella, Sara; Bari, Elia; Colombo, Lino | |
An RGD small-molecule integrin antagonist induces detachment-mediated anoikis in glioma cancer stem cells | 1-gen-2018 | Paolillo, Mayra; Galiazzo, Marisa C.; Daga, Antonio; Ciusani, Emilio; Serra, Massimo; Colombo, Lino; Schinelli, Sergio | |
Synthesis of functionalized 6,5- and 7,5-azabicycloalkane amino acids by metathesis reactions | 1-gen-2019 | Serra, M.; Bernardi, E.; De Lorenzi, E.; Colombo, L. | |
Palladium-catalyzed asymmetric decarboxylative allylation of azlactone enol carbonates: Fast access to enantioenriched α-allyl quaternary amino acids | 1-gen-2019 | Serra, M; Bernardi, E; Marrubini, G; De Lorenzi, E; Colombo, L | |
One-Pot Preparation of Functionalized Azabicyclo[6.3.0]alkanone Amino Acids by Tandem Cross Enyne Metathesis/Ring-Closing Metathesis | 1-gen-2020 | Bernardi, E.; Colombo, L.; De Lorenzi, E.; Carraro, M.; Serra, M. | |
Recent Advances in One-Pot Enyne Metathesis Processes for the Preparation of Biologically and Medicinally Relevant Compounds | 1-gen-2021 | Bernardi, E.; Colombo, L.; Serra, M. | |
Synthesis of Functionalized Proline-Derived Azabicycloalkane Amino Acids and Their Applications in Drug Discovery: Recent Advances | 1-gen-2023 | Serra, M.; Terreni, M.; Bernardi, E.; Colombo, L. |
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