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Molecular Insights into Human Monoamine Oxidase B Inhibition by the Glitazone Antidiabetes Drugs 1-gen-2012 Binda, Claudia; Aldeco, M; Geldenhuys, Wj; Tortorici, Marcello; Mattevi, Andrea; Edmondson, De
Structural Basis for Benzothiazinone-Mediated Killing of Mycobacterium tuberculosis. 1-gen-2012 Neres, J; Pojer, F; Molteni, Elisabetta; Chiarelli, Laurent; Dhar, N; Boy Röttger, S; Buroni, Silvia; Fullam, E; Degiacomi, Giulia; Lucarelli, Ap; Read, Rj; Zanoni, Giuseppe; Edmondson, De; DE ROSSI, Edda; Pasca, MARIA ROSALIA; Mckinney, Jd; Dyson, Pj; Riccardi, Giovanna; Mattevi, Andrea; Cole, St; Binda, Claudia
The DprE1 enzyme, one of the most vulnerable targets of Mycobacterium tuberculosis. 1-gen-2013 Riccardi, Giovanna; Pasca, MARIA ROSALIA; Chiarelli, Laurent; Manina, Giulia; Mattevi, Andrea; Binda, Claudia
4-Aminoquinolone Piperidine Amides: Non-Covalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity. 1-gen-2014 Naik, M; Humnabadkar, V; Tantry, Sj; Panda, M; Narayan, A; Guptha, S; Panduga, V; Manjrekar, P; Jena, Lk; Koushik, K; Shanbhag, G; Jatheendranath, S; M. R., M.; Gorai, G; Bathula, C; Rudrapatna, S; Achar, V; Sharma, S; Ambady, A; Hegde, N; Mahadevaswamy, J; Kaur, P; Sambandamurthy, Vk; Awasthy, D; Narayanan, C; Ravishankar, S; Madhavapeddi, P; Reddy, J; Kr, P; Saralaya, R; Chatterji, M; Whiteaker, J; Mclaughlin, R; Chiarelli, Laurent; Riccardi, Giovanna; Pasca, MARIA ROSALIA; Binda, Claudia; Neres, Jp; Dhar, N; Signorino Gelo, F; Mckinney, J; Ramachandran, V; Shandil, R; Tommasi, R; Iyer, Ps; Narayanan, S; Hosagrahara, V; Kavanagh, S; Dinesh, N; Ghorpade, S. R.
Kinetic and structural analysis of the irreversible inhibition of human monoamine oxidases by ASS234, a multi-target compound designed for use in Alzheimer's disease 1-gen-2014 Esteban, G; Allan, J; Samadi, A; Mattevi, Andrea; Unzeta, M; Marco Contelles, J; Binda, Claudia; Ramsay, R.
Structure-Based Enzyme Tailoring of 5-Hydroxymethylfurfural Oxidase 1-gen-2015 Willem P., Dijkman; Binda, Claudia; Marco W., Fraaije; Mattevi, Andrea
2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1. 1-gen-2015 Neres, J; Hartkoorn, Rc; Chiarelli, Laurent; Gadupudi, R; Pasca, MARIA ROSALIA; Mori, Giorgia; Venturelli, A; Savina, S; Makarov, V; Kolly, Gs; Molteni, E; Binda, Claudia; Dhar, N; Ferrari, S; Brodin, P; Delorme, V; Landry, V; de Jesus Lopes Ribeiro, Al; Farina, D; Saxena, P; Pojer, F; Carta, A; Luciani, R; Porta, Alessio; Zanoni, G; DE ROSSI, Edda; Costi, Mp; Riccardi, Giovanna; Cole, S. T.
An unprecedented NADPH domain conformation in lysine monooxygenase NbtG provides insights into uncoupling of oxygen consumption from substrate hydroxylation 1-gen-2015 Binda, Claudia; Robinson, Reeder M; Martin Del Campo, Julia S; Keul, Nicholas D; Rodriguez, Pedro J; Robinson, Howard H; Mattevi, Andrea; Sobrado, Pablo
Biocatalytic Characterization of Human FMO5: Unearthing Baeyer-Villiger Reactions in Humans 1-gen-2016 Fiorentini, Filippo; Geier, Martina; Binda, Claudia; Winkler, Margit; Faber, Kurt; Hall, Mélanie; Mattevi, Andrea
Design and synthesis of novel chalcones as potent selective monoamine oxidase-B inhibitors. 1-gen-2016 Hammuda, A; Shalaby, R; Rovida, Stefano; Edmondson, De; Binda, Claudia; Khalil, A.
Biocatalytic Properties and Structural Analysis of Eugenol Oxidase from Rhodococcus jostii RHA1: A Versatile Oxidative Biocatalyst 1-gen-2016 Nguyen, QUOC THAI; Degonzalo, Gonzalo; Binda, Claudia; Rioz Martínez, Ana; Mattevi, Andrea; Fraaije, Marco W.
Monoamine Oxidases, Oxidative Stress, and Altered Mitochondrial Dynamics in Cardiac Ageing 1-gen-2017 Maggiorani, D; Manzella, Nicola; Edmondson, De; Mattevi, Andrea; Parini, A; Binda, Claudia; Mialet Perez, J.
Two tyrosine residues, Tyr-108 and Tyr-503, are responsible for the deprotonation of phenolic substrates in vanillyl-alcohol oxidase. 1-gen-2017 Ewing, Ta; Nguyen, QUOC THAI; Allan, Rc; Gygli, G; Romero, E; Binda, Claudia; Fraaije, Mw; Mattevi, Andrea; van Berkel, Wjh
Isolation and characterization of a thermostable F420:NADPH oxidoreductase from Thermobifida fusca 1-gen-2017 Kumar, Hemant; Nguyen, QUOC THAI; Binda, Claudia; Mattevi, Andrea; Fraaije, MARCO WILHELMUS
Discovery and characterization of an F420-dependent glucose-6-phosphate dehydrogenase (Rh-FGD1) from Rhodococcus jostii RHA1 1-gen-2017 Nguyen, QUOC THAI; Trinco, G; Binda, Claudia; Mattevi, Andrea; Fraaije, Mw
Comparative Analysis of the Neurochemical Profile and MAO Inhibition Properties of N‑(Furan-2-ylmethyl)‑N‑methylprop-2-yn-1-amine 1-gen-2017 De Deurwaerdère, P; Binda, Claudia; Corne, R; Leone, C; Valeri, A; Valoti, M; Ramsay, Rr; Fall, Y; Marco Contelles, J.
Monoamine Oxidases 1-gen-2018 Binda, Claudia
Monoamine oxidase-A is a novel driver of stress-induced premature senescence through inhibition of parkin-mediated mitophagy 1-gen-2018 Manzella, Nicola; Santin, Yohan; Maggiorani, Damien; Martini, Hélène; Douin-Echinard, Victorine; Passos, Joao F.; Lezoualc'H, Frank; Binda, Claudia; Parini, Angelo; Mialet-Perez, Jeanne
Tight-Binding Inhibition of Human Monoamine Oxidase B by Chromone Analogs: A Kinetic, Crystallographic, and Biological Analysis 1-gen-2018 COSTA REIS, JOANA ALEXANDRA; Manzella, Nicola; Cagide, Fernando; Mialet-Perez, Jeanne; Uriarte, Eugenio; Parini, Angelo; Borges, Fernanda; Binda, Claudia
Structure-Based Engineering of Phanerochaete chrysosporium Alcohol Oxidase for Enhanced Oxidative Power toward Glycerol 1-gen-2018 Nguyen, QUOC THAI; Romero, Elvira; Dijkman, Willem P.; De Vasconcellos, Suzan Pantaroto; Binda, Claudia; Mattevi, Andrea; Fraaije, MARCO WILHELMUS
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