Sfoglia per Rivista ACS MEDICINAL CHEMISTRY LETTERS
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry.
2020-01-01 Azzali, E; Girardini, M; Annunziato, G; Pavone, M; Vacondio, F; Mori, G; Pasca, Mr; Costantino, G; Pieroni, M.
3D-QSAR-Assisted Design, Synthesis, and Evaluation of Novobiocin Analogues
2013-01-01 Zhao, Huiping; Moroni, Elisabetta; Yan, Bin; Colombo, Giorgio; Blagg, Brian S. J.
BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application
2020-01-01 Della Volpe, S.; Listro, R.; Parafioriti, M.; Di Giacomo, M.; Rossi, D.; Ambrosio, F. A.; Costa, G.; Alcaro, S.; Ortuso, F.; Hirsch, A. K. H.; Vasile, F.; Collina, S.
Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
2023-01-01 Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita
Design, Syntheses, and Anti-TB Activity of 1,3-Benzothiazinone Azide and Click Chemistry Products Inspired by BTZ043
2016-01-01 Tiwari, R.; Miller, P. A.; Chiarelli, Laurent; Mori, Giorgia; Šarkan, M.; Centárová, I.; Cho, S.; Mikušová, K.; Franzblau, S. G.; Oliver, A. G.; Miller, M. J.
Development of 6-Methanesulfonyl-8-nitrobenzothiazinone Based Antitubercular Agents
2022-01-01 Shi, R.; Wang, B.; Stelitano, G.; Wu, X.; Shan, Y.; Wu, Y.; Wang, X.; Chiarelli, L. R.; Lu, Y.; Qiao, C.
Dual Reversible Coumarin Inhibitors Mutually Bound to Monoamine Oxidase B and Acetylcholinesterase Crystal Structures
2022-01-01 Ekstrom, F.; Gottinger, A.; Forsgren, N.; Catto, M.; Iacovino, L. G.; Pisani, L.; Binda, C.
Identification of a New Scaffold for Hsp90 C-Terminal Inhibition
2014-01-01 Zhao, Huiping; Moroni, Elisabetta; Colombo, Giorgio; Blagg, Brian S. J.
Inhibition of β-Amyloid Aggregation in Alzheimer's Disease: The Key Role of (Pro)electrophilic Warheads
2022-01-01 Basagni, F.; Naldi, M.; Ginex, T.; Luque, F. J.; Fagiani, F.; Lanni, C.; Iurlo, M.; Marcaccio, M.; Minarini, A.; Bartolini, M.; Rosini, M.
Interplay of Modified Sialic Acid Inhibitors and the Human Parainfluenza Virus 1 Hemagglutinin-Neuraminidase Active Site
2023-01-01 Rota, Paola; La Rocca, Paolo; Bonfante, Francesco; Pagliari, Matteo; Cirillo, Federica; Piccoli, Marco; Ghiroldi, Andrea; Franco, Valentina; Pappone, Carlo; Allevi, Pietro; Anastasia, Luigi
Mechanisms of Metabolite Amyloid Formation: Computational Studies for Drug Design against Metabolic Disorders
2019-01-01 Meli, M.; Engel, H.; Laor, D.; Gazit, E.; Colombo, G.
Molecular Insights into Human Monoamine Oxidase B Inhibition by the Glitazone Antidiabetes Drugs
2012-01-01 Binda, Claudia; Aldeco, M; Geldenhuys, Wj; Tortorici, Marcello; Mattevi, Andrea; Edmondson, De
Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation
2013-01-01 Stefania, Butini; Margherita, Brindisi; Simone, Brogi; Samuele, Maramai; Egeria, Guarino; Alessandro, Panico; Ashima, Saxena; Ved, Chauhan; Colombo, Raffaella; Verga, Laura; DE LORENZI, Ersilia; Manuela, Bartolini; Vincenza, Andrisano; Ettore, Novellino; Giuseppe, Campiani; Sandra, Gemma
Novel Compounds Targeting the RNA-Binding Protein HuR. Structure-Based Design, Synthesis, and Interaction Studies
2019-01-01 DELLA VOLPE, Serena; Nasti, Rita; Queirolo, Michele; Yagiz Unver, M.; Jumde, Varsha K.; Domling, Alexander; Vasile, Francesca; Potenza, Donatella; Alessandra Ambrosio, Francesca; Costa, Giosué; Alcaro, Stefano; Zucal, Chiara; Provenzani, Alessandro; DI GIACOMO, Marcello; Rossi, Daniela; Hirsch, Anna K. H.; Collina, Simona
Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents
2020-01-01 Franchini, S.; Linciano, P.; Puja, G.; Tait, A.; Borsari, C.; Denora, N.; Iacobazzi, R. M.; Brasili, L.; Sorbi, C.
Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
2023-01-01 Alfano, Ai; Pelliccia, S; Rossino, G; Chianese, O; Summa, V; Collina, S; Brindisi, M
Promising Non-cytotoxic Monosubstituted Chalcones to Target Monoamine Oxidase-B
2021-01-01 Iacovino, L. G.; Pinzi, L.; Facchetti, G.; Bortolini, B.; Christodoulou, M. S.; Binda, C.; Rastelli, G.; Rimoldi, I.; Passarella, D.; Di Paolo, M. L.; Dalla Via, L.
Pure Diastereomers of a Tranylcypromine-Based LSD1 Inhibitor: Enzyme Selectivity and In-Cell Studies
2015-01-01 Valente, S; Rodriguez, V; Mercurio, C; Vianello, P; Saponara, B; Cirilli, R; Ciossani, Giuseppe; Labella, D; Marrocco, B; Ruoppolo, G; Botrugno, Oa; Dessanti, P; Minucci, S; Mattevi, Andrea; Varasi, M; Mai, A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry. | 1-gen-2020 | Azzali, E; Girardini, M; Annunziato, G; Pavone, M; Vacondio, F; Mori, G; Pasca, Mr; Costantino, G; Pieroni, M. | |
| 3D-QSAR-Assisted Design, Synthesis, and Evaluation of Novobiocin Analogues | 1-gen-2013 | Zhao, Huiping; Moroni, Elisabetta; Yan, Bin; Colombo, Giorgio; Blagg, Brian S. J. | |
| BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application | 1-gen-2020 | Della Volpe, S.; Listro, R.; Parafioriti, M.; Di Giacomo, M.; Rossi, D.; Ambrosio, F. A.; Costa, G.; Alcaro, S.; Ortuso, F.; Hirsch, A. K. H.; Vasile, F.; Collina, S. | |
| Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds | 1-gen-2023 | Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita | |
| Design, Syntheses, and Anti-TB Activity of 1,3-Benzothiazinone Azide and Click Chemistry Products Inspired by BTZ043 | 1-gen-2016 | Tiwari, R.; Miller, P. A.; Chiarelli, Laurent; Mori, Giorgia; Šarkan, M.; Centárová, I.; Cho, S.; Mikušová, K.; Franzblau, S. G.; Oliver, A. G.; Miller, M. J. | |
| Development of 6-Methanesulfonyl-8-nitrobenzothiazinone Based Antitubercular Agents | 1-gen-2022 | Shi, R.; Wang, B.; Stelitano, G.; Wu, X.; Shan, Y.; Wu, Y.; Wang, X.; Chiarelli, L. R.; Lu, Y.; Qiao, C. | |
| Dual Reversible Coumarin Inhibitors Mutually Bound to Monoamine Oxidase B and Acetylcholinesterase Crystal Structures | 1-gen-2022 | Ekstrom, F.; Gottinger, A.; Forsgren, N.; Catto, M.; Iacovino, L. G.; Pisani, L.; Binda, C. | |
| Identification of a New Scaffold for Hsp90 C-Terminal Inhibition | 1-gen-2014 | Zhao, Huiping; Moroni, Elisabetta; Colombo, Giorgio; Blagg, Brian S. J. | |
| Inhibition of β-Amyloid Aggregation in Alzheimer's Disease: The Key Role of (Pro)electrophilic Warheads | 1-gen-2022 | Basagni, F.; Naldi, M.; Ginex, T.; Luque, F. J.; Fagiani, F.; Lanni, C.; Iurlo, M.; Marcaccio, M.; Minarini, A.; Bartolini, M.; Rosini, M. | |
| Interplay of Modified Sialic Acid Inhibitors and the Human Parainfluenza Virus 1 Hemagglutinin-Neuraminidase Active Site | 1-gen-2023 | Rota, Paola; La Rocca, Paolo; Bonfante, Francesco; Pagliari, Matteo; Cirillo, Federica; Piccoli, Marco; Ghiroldi, Andrea; Franco, Valentina; Pappone, Carlo; Allevi, Pietro; Anastasia, Luigi | |
| Mechanisms of Metabolite Amyloid Formation: Computational Studies for Drug Design against Metabolic Disorders | 1-gen-2019 | Meli, M.; Engel, H.; Laor, D.; Gazit, E.; Colombo, G. | |
| Molecular Insights into Human Monoamine Oxidase B Inhibition by the Glitazone Antidiabetes Drugs | 1-gen-2012 | Binda, Claudia; Aldeco, M; Geldenhuys, Wj; Tortorici, Marcello; Mattevi, Andrea; Edmondson, De | |
| Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation | 1-gen-2013 | Stefania, Butini; Margherita, Brindisi; Simone, Brogi; Samuele, Maramai; Egeria, Guarino; Alessandro, Panico; Ashima, Saxena; Ved, Chauhan; Colombo, Raffaella; Verga, Laura; DE LORENZI, Ersilia; Manuela, Bartolini; Vincenza, Andrisano; Ettore, Novellino; Giuseppe, Campiani; Sandra, Gemma | |
| Novel Compounds Targeting the RNA-Binding Protein HuR. Structure-Based Design, Synthesis, and Interaction Studies | 1-gen-2019 | DELLA VOLPE, Serena; Nasti, Rita; Queirolo, Michele; Yagiz Unver, M.; Jumde, Varsha K.; Domling, Alexander; Vasile, Francesca; Potenza, Donatella; Alessandra Ambrosio, Francesca; Costa, Giosué; Alcaro, Stefano; Zucal, Chiara; Provenzani, Alessandro; DI GIACOMO, Marcello; Rossi, Daniela; Hirsch, Anna K. H.; Collina, Simona | |
| Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents | 1-gen-2020 | Franchini, S.; Linciano, P.; Puja, G.; Tait, A.; Borsari, C.; Denora, N.; Iacobazzi, R. M.; Brasili, L.; Sorbi, C. | |
| Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds | 1-gen-2023 | Alfano, Ai; Pelliccia, S; Rossino, G; Chianese, O; Summa, V; Collina, S; Brindisi, M | |
| Promising Non-cytotoxic Monosubstituted Chalcones to Target Monoamine Oxidase-B | 1-gen-2021 | Iacovino, L. G.; Pinzi, L.; Facchetti, G.; Bortolini, B.; Christodoulou, M. S.; Binda, C.; Rastelli, G.; Rimoldi, I.; Passarella, D.; Di Paolo, M. L.; Dalla Via, L. | |
| Pure Diastereomers of a Tranylcypromine-Based LSD1 Inhibitor: Enzyme Selectivity and In-Cell Studies | 1-gen-2015 | Valente, S; Rodriguez, V; Mercurio, C; Vianello, P; Saponara, B; Cirilli, R; Ciossani, Giuseppe; Labella, D; Marrocco, B; Ruoppolo, G; Botrugno, Oa; Dessanti, P; Minucci, S; Mattevi, Andrea; Varasi, M; Mai, A. |
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