Sfoglia per Autore
Ureidopyridazine derivatives as Acyl-CoA:cholesterol acyltransferase inhibitors
2006-01-01 Gelain, Arianna; Bettinelli, Ilaria; Barlocco, Daniela; KWON Byoung, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio
3-Heptylamino-5-phenylpyridazine derivatives as analogues of acyl-CoA: cholesterol acyltransferase inhibitors containing the N-heptyl-N’-arylureidic moiety
2006-01-01 Gelain, Arianna; Barlocco, Daniela; KWON Byong, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio
Synthesis, conformational studies, binding assessment and liposome insertion of a thioether-bridged mimetic of the antigen GM3 ganglioside lactone
2007-01-01 Toma, Lucio; Di Cola, Emanuela; Ienco, Andrea; Legnani, Laura; Lunghi, Carlotta; Moneti, Gloriano; Richichi, Barbara; Ristori, Sandra; Dell'Atti, Daniela; Nativi, Cristina
Alternative mechanistic paths in the hetero-Diels-Alder reaction of alpha-oxothiones: a theoretical study
2007-01-01 Legnani, Laura; Lunghi, Carlotta; Marinone, Franca; Nativi, Cristina; Richichi, Barbara; Toma, Lucio
A full conformational characterization of 13-ethylprogestogens through theoretical calculations and nuclear magnetic resonance spectroscopy
2007-01-01 Colombo, Diego; Ferraboschi, Patrizia; Legnani, Laura; Prestileo, Paolo; Toma, Lucio
A new stereoselective approach to a selectively protected derivative of D-pinitol and its evaluation as alpha-L-rhamnopyranose mimetic
2008-01-01 Catelani, Giorgio; D'Andrea, Felicia; Griselli, Alessio; Guazzelli, Lorenzo; Legnani, Laura; Toma, Lucio
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors
2008-01-01 Murineddu, Gabriele; Murruzzu, Caterina; Curzu Maria, M; Chelucci, Giorgio; Gotti, Cecilia; Gaimarri, Annalisa; Legnani, Laura; Toma, Lucio; Pinna Gerard, A.
Complete 1H and 13C assignments of (21R) and (21S) diastereomers of argatroban
2008-01-01 Colombo, Diego; Ferraboschi, Patrizia; Grisenti, Paride; Legnani, Laura
A full conformational characterization of natural ionones and irones, as well as 13-alkyl-substituted alpha-ionones
2008-01-01 Legnani, Laura; Luparia, Marco; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni
Biphenyl versus Phenylpyridazine Derivatives: The Role of the Heterocycle in a Series of Acyl-CoA:Cholesterol Acyl Transferase Inhibitors
2008-01-01 Gelain, Arianna; Barlocco, Daniela; Kwon Byoung, Mog; Jeong Tae, Sook; Im Kyung, Ran; Legnani, Laura; Toma, Lucio
Enantioselective Synthesis and Olfactory Evaluation of Bicyclic r- andγ-Ionone Derivatives: The 3D Arrangement of Key Molecular FeaturesRelevant to the Violet Odor of Ionones
2009-01-01 Luparia, Marco; Legnani, Laura; Porta, Alessio; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni
Synthesis, molecular dynamics simulations, and biology of a carba-analogue of the trisaccharide repeating unit of Streptococcus pneumoniae 19F capsular polysaccharide
2009-01-01 Legnani, Laura; Ronchi, Silvia; Fallarini, Silvia; Lombardi, Grazia; Campo, Federica; Panza, Luigi; Lay, Luigi; Poletti, Laura; Toma, Lucio; Ronchetti, Fiamma; Compostella, Federica
An exhaustive conformational evaluation of the HIV-1 inhibitor BMS-378806 through theoretical calculations and nuclear magnetic resonance spectroscopy
2009-01-01 Colombo, Diego; Villa, Stefania; Solano, Lucrezia; Legnani, Laura; Marinone, Franca; Toma, Lucio
Cyclic glycopeptidomimetics through a versatile sugar-based scaffold
2009-01-01 Altamura, Maria; Dragoni, Elisa; Infantino Angela, Simona; Legnani, Laura; Ludbrook Steve, B.; Menchi, Gloria; Toma, Lucio; Nativi, Cristina
Modeling of synthetic phosphono and carba analogues ofN-acetyl-alpha-D-mannosamine 1-phosphate, the repeating unit of the capsular polysaccharide from Neisseria meningitidis serovar A
2009-01-01 Toma, Lucio; Legnani, Laura; Rencurosi, Anna; Poletti, Laura; Lay, Luigi; Russo, Giovanni
Synthesis, modeling, and crystallographic study of 3,4-disubstituted-1,2,5-oxadiazoles and evaluation of their ability to decrease STAT3 activity
2010-01-01 Shin Dae, Seop; Masciocchi, Daniela; Gelain, Arianna; Villa, Stefania; Barlocco, Daniela; Meneghetti, Fiorella; Pedretti, Alessandro; Han Young, Min; Han Dong, Cho; Kwon Byoung, Mog; Legnani, Laura; Toma, Lucio
Stable GM3 Lactone Mimetic Raises Antibodies Specific for the Antigens Expressed on Melanoma Cells
2010-01-01 Arcangeli, Annarosa; Toma, Lucio; Contiero, Luca; Crociani, Olivia; Legnani, Laura; Lunghi, Carlotta; Nesti, Elisa; Moneti, Gloriano; Richichi, Barbara; Nativi, Cristina
Modeling and Spectroscopic Studies of Synthetic Diazabicyclo Analogs of the HIV-1 Inhibitor BMS-378806 and Evaluation of Their Antiviral Activity
2011-01-01 Legnani, Laura; Colombo, Diego; Cocchi, Elena; Solano, Lucrezia; Villa, Stefania; Lopalco, Lucia; Asti, Valeria; Diomede, Lorenzo; Marinone, Franca; Toma, Lucio
Molecular dynamics simulations of the Salmonella typhi Vi antigenic polysaccharide and effects of the introduction of a zwitterionic motif
2011-01-01 Legnani, Laura; Compostella, Federica; Grazioso, Giovanni; Marinone, Franca; Toma, Lucio
Mechanism of falcipain-2 inhibition by a,b-unsaturated benzo[1,4]diazepin-2-one methyl ester
2012-01-01 Grazioso, G.; Legnani, Laura; Toma, Lucio; Ettari, R.; Micale, N.; De Micheli, C.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Ureidopyridazine derivatives as Acyl-CoA:cholesterol acyltransferase inhibitors | 1-gen-2006 | Gelain, Arianna; Bettinelli, Ilaria; Barlocco, Daniela; KWON Byoung, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio | |
3-Heptylamino-5-phenylpyridazine derivatives as analogues of acyl-CoA: cholesterol acyltransferase inhibitors containing the N-heptyl-N’-arylureidic moiety | 1-gen-2006 | Gelain, Arianna; Barlocco, Daniela; KWON Byong, Mog; JEONG Tae, Sook; IM Kyung, Ran; Legnani, Laura; Toma, Lucio | |
Synthesis, conformational studies, binding assessment and liposome insertion of a thioether-bridged mimetic of the antigen GM3 ganglioside lactone | 1-gen-2007 | Toma, Lucio; Di Cola, Emanuela; Ienco, Andrea; Legnani, Laura; Lunghi, Carlotta; Moneti, Gloriano; Richichi, Barbara; Ristori, Sandra; Dell'Atti, Daniela; Nativi, Cristina | |
Alternative mechanistic paths in the hetero-Diels-Alder reaction of alpha-oxothiones: a theoretical study | 1-gen-2007 | Legnani, Laura; Lunghi, Carlotta; Marinone, Franca; Nativi, Cristina; Richichi, Barbara; Toma, Lucio | |
A full conformational characterization of 13-ethylprogestogens through theoretical calculations and nuclear magnetic resonance spectroscopy | 1-gen-2007 | Colombo, Diego; Ferraboschi, Patrizia; Legnani, Laura; Prestileo, Paolo; Toma, Lucio | |
A new stereoselective approach to a selectively protected derivative of D-pinitol and its evaluation as alpha-L-rhamnopyranose mimetic | 1-gen-2008 | Catelani, Giorgio; D'Andrea, Felicia; Griselli, Alessio; Guazzelli, Lorenzo; Legnani, Laura; Toma, Lucio | |
Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors | 1-gen-2008 | Murineddu, Gabriele; Murruzzu, Caterina; Curzu Maria, M; Chelucci, Giorgio; Gotti, Cecilia; Gaimarri, Annalisa; Legnani, Laura; Toma, Lucio; Pinna Gerard, A. | |
Complete 1H and 13C assignments of (21R) and (21S) diastereomers of argatroban | 1-gen-2008 | Colombo, Diego; Ferraboschi, Patrizia; Grisenti, Paride; Legnani, Laura | |
A full conformational characterization of natural ionones and irones, as well as 13-alkyl-substituted alpha-ionones | 1-gen-2008 | Legnani, Laura; Luparia, Marco; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni | |
Biphenyl versus Phenylpyridazine Derivatives: The Role of the Heterocycle in a Series of Acyl-CoA:Cholesterol Acyl Transferase Inhibitors | 1-gen-2008 | Gelain, Arianna; Barlocco, Daniela; Kwon Byoung, Mog; Jeong Tae, Sook; Im Kyung, Ran; Legnani, Laura; Toma, Lucio | |
Enantioselective Synthesis and Olfactory Evaluation of Bicyclic r- andγ-Ionone Derivatives: The 3D Arrangement of Key Molecular FeaturesRelevant to the Violet Odor of Ionones | 1-gen-2009 | Luparia, Marco; Legnani, Laura; Porta, Alessio; Zanoni, Giuseppe; Toma, Lucio; Vidari, Giovanni | |
Synthesis, molecular dynamics simulations, and biology of a carba-analogue of the trisaccharide repeating unit of Streptococcus pneumoniae 19F capsular polysaccharide | 1-gen-2009 | Legnani, Laura; Ronchi, Silvia; Fallarini, Silvia; Lombardi, Grazia; Campo, Federica; Panza, Luigi; Lay, Luigi; Poletti, Laura; Toma, Lucio; Ronchetti, Fiamma; Compostella, Federica | |
An exhaustive conformational evaluation of the HIV-1 inhibitor BMS-378806 through theoretical calculations and nuclear magnetic resonance spectroscopy | 1-gen-2009 | Colombo, Diego; Villa, Stefania; Solano, Lucrezia; Legnani, Laura; Marinone, Franca; Toma, Lucio | |
Cyclic glycopeptidomimetics through a versatile sugar-based scaffold | 1-gen-2009 | Altamura, Maria; Dragoni, Elisa; Infantino Angela, Simona; Legnani, Laura; Ludbrook Steve, B.; Menchi, Gloria; Toma, Lucio; Nativi, Cristina | |
Modeling of synthetic phosphono and carba analogues ofN-acetyl-alpha-D-mannosamine 1-phosphate, the repeating unit of the capsular polysaccharide from Neisseria meningitidis serovar A | 1-gen-2009 | Toma, Lucio; Legnani, Laura; Rencurosi, Anna; Poletti, Laura; Lay, Luigi; Russo, Giovanni | |
Synthesis, modeling, and crystallographic study of 3,4-disubstituted-1,2,5-oxadiazoles and evaluation of their ability to decrease STAT3 activity | 1-gen-2010 | Shin Dae, Seop; Masciocchi, Daniela; Gelain, Arianna; Villa, Stefania; Barlocco, Daniela; Meneghetti, Fiorella; Pedretti, Alessandro; Han Young, Min; Han Dong, Cho; Kwon Byoung, Mog; Legnani, Laura; Toma, Lucio | |
Stable GM3 Lactone Mimetic Raises Antibodies Specific for the Antigens Expressed on Melanoma Cells | 1-gen-2010 | Arcangeli, Annarosa; Toma, Lucio; Contiero, Luca; Crociani, Olivia; Legnani, Laura; Lunghi, Carlotta; Nesti, Elisa; Moneti, Gloriano; Richichi, Barbara; Nativi, Cristina | |
Modeling and Spectroscopic Studies of Synthetic Diazabicyclo Analogs of the HIV-1 Inhibitor BMS-378806 and Evaluation of Their Antiviral Activity | 1-gen-2011 | Legnani, Laura; Colombo, Diego; Cocchi, Elena; Solano, Lucrezia; Villa, Stefania; Lopalco, Lucia; Asti, Valeria; Diomede, Lorenzo; Marinone, Franca; Toma, Lucio | |
Molecular dynamics simulations of the Salmonella typhi Vi antigenic polysaccharide and effects of the introduction of a zwitterionic motif | 1-gen-2011 | Legnani, Laura; Compostella, Federica; Grazioso, Giovanni; Marinone, Franca; Toma, Lucio | |
Mechanism of falcipain-2 inhibition by a,b-unsaturated benzo[1,4]diazepin-2-one methyl ester | 1-gen-2012 | Grazioso, G.; Legnani, Laura; Toma, Lucio; Ettari, R.; Micale, N.; De Micheli, C. |
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