Sfoglia per Autore
Synthesis and in vitro evaluation of novel pan-SR modulators: Identification of (E)-4-benzyl-1-[3-(naphthalen-2-yl)but-2-en-1-yl]piperidine (RC-106) as potential anticancer agent.
2016-01-01 Rui, Marta; Rossi, Daniela; Marra, Annamaria; Paolillo, Mayra; Curti, Daniela; Tesei, A; Cortesi, Michela; Pace, V; Collina, Simona
“Fit-for-purpose” development of analytical and (semi)preparative enantioselective high performance liquid and supercritical fluid chromatography for the access to a novel sigma1 receptor agonist.
2016-01-01 Rossi, Daniela; Marra, Annamaria; Rui, Marta; Brambilla, Stefania; Juza, Markus; Collina, Simona
Toward the identification of neuroprotective agents: G-scale synthesis, pharmacokinetic evaluation and CNS distribution of (R)-RC-33, a promising SIGMA1 receptor agonist
2016-01-01 Marra, Annamaria; Rossi, Daniela; Pignataro, L.; Bigogno, C.; Canta, A.; Oggioni, N.; Malacrida, A. .; Corbo, M.; Cavaletti, G.; Peviani, Marco; Curti, Daniela; Dondio, G.; Collina, Simona
Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A3 Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy
2016-01-01 Rossi, Daniela; Nasti, Rita; Marra, Annamaria; Meneghini, Silvia; Mazzeo, G.; Longhi, G.; Memo, M.; Cosimelli, B.; Greco, G.; Novellino, E.; Da Settimo, F.; Martini, C.; Taliani, S.; Abbate, S.; Collina, Simona
Novel enantiopure sigma receptor modulators: Quick (semi-)preparative chiral resolution via hplc and absolute configuration assignment
2016-01-01 Rui, Marta; Marra, Annamaria; Pace, V.; Juza, M.; Rossi, Daniela; Collina, Simona
Development of easy-to-use reverse-phase liquid chromatographic methods for determining PRE-084, RC-33 and RC-34 in biological matrices. The first step for in vivo analysis of sigma1 receptor agonists.
2016-01-01 Marra, Annamaria; Rossi, Daniela; Maggi, Lauretta; Corana, Federica; Mannucci, Barbara; Peviani, Marco; Curti, Daniela; Collina, Simona
Synthesis and biological evaluation of new aryl-alkyl(alkenyl)-4-benzylpiperidines, novel Sigma Receptor (SR) modulators, as potential anticancer-agents
2016-01-01 Rui, Marta; Rossi, Daniela; Marra, Annamaria; Paolillo, Mayra; Schinelli, Sergio; Curti, Daniela; Tesei, A.; Cortesi, M.; Zamagni, A.; Laurini, E.; Pricl, S.; Schepmann, D.; Wűnsch, B.; Urban, E.; Pace, V.; Collina, Simona
Sigma Receptors: Novel Targets For The Treatment Of Highly Malignant Tumors
2017-01-01 Cortesi, Michela; Pignatta, Sara; Collina, Simona; Rui, Marta; Marra, Annamaria; Tosatto, Luigino; Bartolini, Daniela; Nigrisoli, Evandro; Arienti, Andrea Rocca Alice Zamagni Chiara; Zanoni, Michele; Tesei, Anna
PAN-SIGMA RECEPTOR MODULATORS AS PROMISING ANTICANCER-AGENTS. THE STORY OF RC-106
2017-01-01 Rui, Marta; Rossi, Daniela; Marra, Annamaria; Dondio, Giulio; Tesei, A.; Cortesi, Michela; Collina, Simona
Anti-tumor efficacy assessment of the sigma receptor pan modulator RC-106. A promising therapeutic tool for pancreatic cancer
2019-01-01 Tesei, A.; Cortesi, M.; Pignatta, S.; Arienti, C.; Massimo Dondio, G.; Bigogno, C.; Malacrida, A.; Miloso, M.; Meregalli, C.; Chiorazzi, A.; Carozzi, V.; Cavaletti, G.; Rui, M.; Marra, A.; Rossi, D.; Collina, S.
Sigma receptor and aquaporin modulators: chiral resolution, configurational assignment, and preliminary biological profile of RC752 enantiomers
2024-01-01 Listro, Roberta; Marra, Annamaria; Cavalloro, Valeria; Rossino, Giacomo; Linciano, Pasquale; Rossi, Daniela; Casali, Emanuele; De Amici, Marco; Mazzeo, Giuseppe; Longhi, Giovanna; Fusè, Marco; Dondio, Giulio; Pellavio, Giorgia; Laforenza, Umberto; Schepmann, Dirk; Wünsch, Bernhard; Collina, Simona
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and in vitro evaluation of novel pan-SR modulators: Identification of (E)-4-benzyl-1-[3-(naphthalen-2-yl)but-2-en-1-yl]piperidine (RC-106) as potential anticancer agent. | 1-gen-2016 | Rui, Marta; Rossi, Daniela; Marra, Annamaria; Paolillo, Mayra; Curti, Daniela; Tesei, A; Cortesi, Michela; Pace, V; Collina, Simona | |
“Fit-for-purpose” development of analytical and (semi)preparative enantioselective high performance liquid and supercritical fluid chromatography for the access to a novel sigma1 receptor agonist. | 1-gen-2016 | Rossi, Daniela; Marra, Annamaria; Rui, Marta; Brambilla, Stefania; Juza, Markus; Collina, Simona | |
Toward the identification of neuroprotective agents: G-scale synthesis, pharmacokinetic evaluation and CNS distribution of (R)-RC-33, a promising SIGMA1 receptor agonist | 1-gen-2016 | Marra, Annamaria; Rossi, Daniela; Pignataro, L.; Bigogno, C.; Canta, A.; Oggioni, N.; Malacrida, A. .; Corbo, M.; Cavaletti, G.; Peviani, Marco; Curti, Daniela; Dondio, G.; Collina, Simona | |
Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A3 Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy | 1-gen-2016 | Rossi, Daniela; Nasti, Rita; Marra, Annamaria; Meneghini, Silvia; Mazzeo, G.; Longhi, G.; Memo, M.; Cosimelli, B.; Greco, G.; Novellino, E.; Da Settimo, F.; Martini, C.; Taliani, S.; Abbate, S.; Collina, Simona | |
Novel enantiopure sigma receptor modulators: Quick (semi-)preparative chiral resolution via hplc and absolute configuration assignment | 1-gen-2016 | Rui, Marta; Marra, Annamaria; Pace, V.; Juza, M.; Rossi, Daniela; Collina, Simona | |
Development of easy-to-use reverse-phase liquid chromatographic methods for determining PRE-084, RC-33 and RC-34 in biological matrices. The first step for in vivo analysis of sigma1 receptor agonists. | 1-gen-2016 | Marra, Annamaria; Rossi, Daniela; Maggi, Lauretta; Corana, Federica; Mannucci, Barbara; Peviani, Marco; Curti, Daniela; Collina, Simona | |
Synthesis and biological evaluation of new aryl-alkyl(alkenyl)-4-benzylpiperidines, novel Sigma Receptor (SR) modulators, as potential anticancer-agents | 1-gen-2016 | Rui, Marta; Rossi, Daniela; Marra, Annamaria; Paolillo, Mayra; Schinelli, Sergio; Curti, Daniela; Tesei, A.; Cortesi, M.; Zamagni, A.; Laurini, E.; Pricl, S.; Schepmann, D.; Wűnsch, B.; Urban, E.; Pace, V.; Collina, Simona | |
Sigma Receptors: Novel Targets For The Treatment Of Highly Malignant Tumors | 1-gen-2017 | Cortesi, Michela; Pignatta, Sara; Collina, Simona; Rui, Marta; Marra, Annamaria; Tosatto, Luigino; Bartolini, Daniela; Nigrisoli, Evandro; Arienti, Andrea Rocca Alice Zamagni Chiara; Zanoni, Michele; Tesei, Anna | |
PAN-SIGMA RECEPTOR MODULATORS AS PROMISING ANTICANCER-AGENTS. THE STORY OF RC-106 | 1-gen-2017 | Rui, Marta; Rossi, Daniela; Marra, Annamaria; Dondio, Giulio; Tesei, A.; Cortesi, Michela; Collina, Simona | |
Anti-tumor efficacy assessment of the sigma receptor pan modulator RC-106. A promising therapeutic tool for pancreatic cancer | 1-gen-2019 | Tesei, A.; Cortesi, M.; Pignatta, S.; Arienti, C.; Massimo Dondio, G.; Bigogno, C.; Malacrida, A.; Miloso, M.; Meregalli, C.; Chiorazzi, A.; Carozzi, V.; Cavaletti, G.; Rui, M.; Marra, A.; Rossi, D.; Collina, S. | |
Sigma receptor and aquaporin modulators: chiral resolution, configurational assignment, and preliminary biological profile of RC752 enantiomers | 1-gen-2024 | Listro, Roberta; Marra, Annamaria; Cavalloro, Valeria; Rossino, Giacomo; Linciano, Pasquale; Rossi, Daniela; Casali, Emanuele; De Amici, Marco; Mazzeo, Giuseppe; Longhi, Giovanna; Fusè, Marco; Dondio, Giulio; Pellavio, Giorgia; Laforenza, Umberto; Schepmann, Dirk; Wünsch, Bernhard; Collina, Simona |
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