ROSSINO, GIACOMO

ROSSINO, GIACOMO  

DIPARTIMENTO DI SCIENZE DEL FARMACO  

Mostra records
Risultati 1 - 20 di 22 (tempo di esecuzione: 0.126 secondi).
Titolo Data di pubblicazione Autore(i) File
Approaches for multi-gram scale isolation of enantiomers for drug discovery 1-gen-2017 Rossi, D.; Tarantino, M.; Rossino, G.; Rui, M.; Juza, M.; Collina, S.
Biocatalysis: A smart and green tool for the preparation of chiral drugs 1-gen-2022 Rossino, G; Robescu, Ms; Licastro, E; Tedesco, C; Martello, I; Maffei, L; Vincenti, G; Bavaro, T; Collina, S
Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization 1-gen-2021 Rossino, G.; Rui, M.; Linciano, P.; Rossi, D.; Boiocchi, M.; Peviani, M.; Poggio, E.; Curti, D.; Schepmann, D.; Wünsch, B.; González-Avendaño, M.; Vergara-Jaque, A.; Caballero, J.; Collina, S.
CHAPTER 12: Sigma Receptors as New Target for Multiple Sclerosis 1-gen-2019 Rui, M.; Rossino, G.; Rossi, D.; Collina, S.
Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds 1-gen-2023 Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita
Enantiomeric Resolution and Absolute Configuration of a Chiral δ-Lactam, Useful Intermediate for the Synthesis of Bioactive Compounds 1-gen-2020 Listro, R; Rossino, G.; Della Volpe, S.; Stabile, R.; Boiocchi, M.; Malavasi, L.; Rossi, D.; Collina, S.
Exploring the RC-106 Chemical Space: Design and Synthesis of Novel (E)-1-(3-Arylbut-2-en-1-yl)-4-(Substituted) Piperazine Derivatives as Potential Anticancer Agents. 1-gen-2020 Listro, R.; Stotani, S.; Rossino, G.; Rui, M.; Malacrida, A.; Cavaletti, G.; Cortesi, M.; Arienti, C.; Tesei, A.; Rossi, D.; Di Giacomo, M.; Miloso, M.; Collina, S.
From Nature to Synthetic Compounds: Novel 1(N),2,3 Trisubstituted-5-oxopyrrolidines Targeting Multiple Myeloma Cells 1-gen-2022 Listro, Roberta; Malacrida, Alessio; Ambrosio, Francesca Alessandra; Rossino, Giacomo; Di Giacomo, Marcello; Cavalloro, Valeria; Garbagnoli, Martina; Linciano, Pasquale; Rossi, Daniela; Cavaletti, Guido; Costa, Giosuè; Alcaro, Stefano; Miloso, Mariarosaria; Collina, Simona
Identification of dual Sigma1 receptor modulators/acetylcholinesterase inhibitors with antioxidant and neurotrophic properties, as neuroprotective agents 1-gen-2018 Rui, Marta; Rossino, Giacomo; Coniglio, Stefania; Monteleone, Stefania; Scuteri, Arianna; Malacrida, Alessio; Rossi, Daniela; Catenacci, Laura; Sorrenti, Milena; Paolillo, Mayra; Curti, Daniela; Venturini, Letizia; Schepmann, Dirk; Wünsch, Bernhard; Liedl, Klaus R.; Cavaletti, Guido; Pace, Vittorio; Urban, Ernst; Collina, Simona
New Insights into the Opening of the Occluded Ligand-Binding Pocket of Sigma1 Receptor: Binding of a Novel Bivalent RC-33 Derivative 1-gen-2020 Rossino, G.; Orellana, I.; Caballero, J.; Schepmann, D.; Wunsch, B.; Rui, M.; Rossi, D.; Gonzalez-Avendano, M.; Collina, S.; Vergara-Jaque, A.
Novel S1R agonists counteracting NMDA excitotoxicity and oxidative stress: A step forward in the discovery of neuroprotective agents 1-gen-2023 Linciano, Pasquale; Sorbi, Claudia; Rossino, Giacomo; Rossi, Daniela; Marsala, Andrea; Denora, Nunzio; Bedeschi, Martina; Marino, Noemi; Miserocchi, Giacomo; Dondio, Giulio; Peviani, Marco; Tesei, Anna; Collina, Simona; Franchini, Silvia
PEG 400/cerium ammonium nitrate combined with microwave-assisted synthesis for rapid access to beta-amino ketones. an easy-to-use protocol for discovering new hit compounds 1-gen-2018 Rossino, Giacomo; Raimondi, M. V.; Rui, M.; Di Giacomo, M.; Rossi, D.; Collina, S.
Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds 1-gen-2023 Alfano, Ai; Pelliccia, S; Rossino, G; Chianese, O; Summa, V; Collina, S; Brindisi, M
PKC in regenerative therapy: New insights for old targets 1-gen-2017 Rui, Marta; Nasti, Rita; Bignardi, Emanuele; DELLA VOLPE, Serena; Rossino, Giacomo; Rossi, Daniela; Collina, Simona
Repurposing the Antiplatelet Agent Ticlopidine to Counteract the Acute Phase of ER Stress Condition: An Opportunity for Fighting Coronavirus Infections and Cancer 1-gen-2022 Tesei, Anna; Cortesi, Michela; Bedeschi, Martina; Marino, Noemi; Rossino, Giacomo; Listro, Roberta; Rossi, Daniela; Linciano, Pasquale; Collina, Simona
Setup and Validation of a Reliable Docking Protocol for the Development of Neuroprotective Agents by Targeting the Sigma-1 Receptor (S1R) 1-gen-2020 Rossino, Giacomo; Rui, Marta; Pozzetti, Luca; Schepmann, Dirk; Wünsch, Bernhard; Zampieri, Daniele; Pellavio, Giorgia; Laforenza, Umberto; Rinaldi, Silvia; Colombo, Giorgio; Morelli, Laura; Linciano, Pasquale; Rossi, Daniela; Collina, Simona
SIGMA 1 RECEPTOR (S1R) MODULATORS AS A THERAPEUTIC STRATEGY FOR PROMOTING NEUROPLASTICITY. DESIGN AND SYNTHESIS OF NOVEL MONO- AND BI-VALENT LIGANDS FOR SRS 20-feb-2020 Rossino, Giacomo
Sigma receptor and aquaporin modulators: chiral resolution, configurational assignment, and preliminary biological profile of RC752 enantiomers 1-gen-2024 Listro, Roberta; Marra, Annamaria; Cavalloro, Valeria; Rossino, Giacomo; Linciano, Pasquale; Rossi, Daniela; Casali, Emanuele; De Amici, Marco; Mazzeo, Giuseppe; Longhi, Giovanna; Fusè, Marco; Dondio, Giulio; Pellavio, Giorgia; Laforenza, Umberto; Schepmann, Dirk; Wünsch, Bernhard; Collina, Simona
Sigma-1 receptor agonists acting on aquaporin-mediated h2o2 permeability: New tools for counteracting oxidative stress 1-gen-2021 Pellavio, G.; Rossino, G.; Gastaldi, G.; Rossi, D.; Linciano, P.; Collina, S.; Laforenza, U.
Sigma-1 receptor antagonists: promising players in fighting neuropathic pain 1-gen-2020 Linciano, Pasquale; Rossino, Giacomo; Listro, Roberta; Rossi, Daniela; Collina, Simona