LINCIANO, PASQUALE
LINCIANO, PASQUALE
DIPARTIMENTO DI SCIENZE DEL FARMACO
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity
2019-01-01 Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L.
4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases
2020-01-01 Linciano, Pasquale; Gianquinto, Eleonora; Montanari, Martina; Maso, Lorenzo; Bellio, Pierangelo; Cebrián-Sastre, Esmeralda; Celenza, Giuseppe; Blázquez, Jesús; Cendron, Laura; Spyrakis, Francesca; Tondi, Donatella
A multidisciplinary approach to the design of novel inhibitors for KPC-2
2017-01-01 Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella
A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol
2019-01-01 Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G.
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
2019-01-01 Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz
An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases
2016-01-01 Quotadamo, Antonio; Linciano, Pasquale; Davoli, Paolo; Tondi, Donatella; Costi, Maria Paola; Venturelli, Alberto
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog
2019-01-01 Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G.
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections
2018-01-01 Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola
Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization
2021-01-01 Rossino, G.; Rui, M.; Linciano, P.; Rossi, D.; Boiocchi, M.; Peviani, M.; Poggio, E.; Curti, D.; Schepmann, D.; Wünsch, B.; González-Avendaño, M.; Vergara-Jaque, A.; Caballero, J.; Collina, S.
Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry
2019-01-01 Citti, C.; Linciano, P.; Panseri, S.; Vezzalini, F.; Forni, F.; Vandelli, M. A.; Cannazza, G.
Chemical and spectroscopic characterization data of ‘cannabidibutol’, a novel cannabidiol butyl analog
2019-01-01 Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G.
Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies
2022-01-01 Linciano, P.; Nasti, R.; Listro, R.; Amadio, M.; Pascale, A.; Potenza, D.; Vasile, F.; Minneci, M.; Ann, J.; Lee, J.; Zhou, X.; Mitchell, G. A.; Blumberg, P. M.; Rossi, D.; Collina, S.
COMPOSTI AD ATTIVITÀ ANTIPARASSITARIA
2019-01-01 Paola Costi, Maria; Costantino, Luca; Linciano, Pasquale; Ferrari, Stefania; Cordeiro da Silva, Anabela
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients?
2023-01-01 D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona
Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth
2019-01-01 Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D’Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Paola Costi, Maria
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
2022-01-01 Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo-Ahen, Outi M H; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela; Giovannetti, Elisa; Peters, Godefridus J; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M; Wade, Rebecca C; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola
Development of therapeutic agents blocking SOS activation
2019-01-01 Maso, L.; Bellio, P.; Linciano, P.; D' Acunto, M.; Celenza, G.; Tondi, Donatella; Cendron, L.
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics
2019-01-01 Borsari, Chiara; Dolores Jimenez-Anton, María; Eick, Julia; Bifeld, Eugenia; Jose Torrado, Juan; Isabel Olías-Molero, Ana; Jesús Corral, María; Santarem, Nuno; Baptista, Catarina; Severi, Leda; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Luciani, Rosaria; Tejera Nevado, Paloma; Zander-Dinse, Dorothea; Franco, Caio H.; Ferrari, Stefania; Moraes, Carolina B.; Cordeiro-da-Silva, Anabela; Ponterini, Glauco; Clos, Joachim; María Alunda, Jose; Paola Costi, Maria
Druggability profile of stilbene-derived PPAR agonists: Determination of physicochemical properties and PAMPA study
2019-01-01 Linciano, P.; De Filippis, B.; Ammazzalorso, A.; Amoia, P.; Cilurzo, F.; Fantacuzzi, M.; Giampietro, L.; Maccallini, C.; Petit, C.; Amoroso, R.
Effect of stilbene and chalcone scaffolds incorporation in clofibric acid on PPARα agonistic activity
2014-01-01 Giampietro, Letizia; D'Angelo, Alessandra; Giancristofaro, Antonella; Ammazzalorso, Alessandra; DE FILIPPIS, Barbara; DI MATTEO, Mauro; Fantacuzzi, Marialuigia; Linciano, Pasquale; Maccallini, Cristina; Amoroso, Rosa
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity | 1-gen-2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L. | |
| 4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases | 1-gen-2020 | Linciano, Pasquale; Gianquinto, Eleonora; Montanari, Martina; Maso, Lorenzo; Bellio, Pierangelo; Cebrián-Sastre, Esmeralda; Celenza, Giuseppe; Blázquez, Jesús; Cendron, Laura; Spyrakis, Francesca; Tondi, Donatella | |
| A multidisciplinary approach to the design of novel inhibitors for KPC-2 | 1-gen-2017 | Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella | |
| A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol | 1-gen-2019 | Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G. | |
| Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform | 1-gen-2019 | Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz | |
| An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases | 1-gen-2016 | Quotadamo, Antonio; Linciano, Pasquale; Davoli, Paolo; Tondi, Donatella; Costi, Maria Paola; Venturelli, Alberto | |
| Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog | 1-gen-2019 | Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G. | |
| Aryl thiosemicarbazones for the treatment of trypanosomatidic infections | 1-gen-2018 | Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola | |
| Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization | 1-gen-2021 | Rossino, G.; Rui, M.; Linciano, P.; Rossi, D.; Boiocchi, M.; Peviani, M.; Poggio, E.; Curti, D.; Schepmann, D.; Wünsch, B.; González-Avendaño, M.; Vergara-Jaque, A.; Caballero, J.; Collina, S. | |
| Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry | 1-gen-2019 | Citti, C.; Linciano, P.; Panseri, S.; Vezzalini, F.; Forni, F.; Vandelli, M. A.; Cannazza, G. | |
| Chemical and spectroscopic characterization data of ‘cannabidibutol’, a novel cannabidiol butyl analog | 1-gen-2019 | Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G. | |
| Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies | 1-gen-2022 | Linciano, P.; Nasti, R.; Listro, R.; Amadio, M.; Pascale, A.; Potenza, D.; Vasile, F.; Minneci, M.; Ann, J.; Lee, J.; Zhou, X.; Mitchell, G. A.; Blumberg, P. M.; Rossi, D.; Collina, S. | |
| COMPOSTI AD ATTIVITÀ ANTIPARASSITARIA | 1-gen-2019 | Paola Costi, Maria; Costantino, Luca; Linciano, Pasquale; Ferrari, Stefania; Cordeiro da Silva, Anabela | |
| Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? | 1-gen-2023 | D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona | |
| Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth | 1-gen-2019 | Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D’Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Paola Costi, Maria | |
| Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth | 1-gen-2022 | Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo-Ahen, Outi M H; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela; Giovannetti, Elisa; Peters, Godefridus J; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M; Wade, Rebecca C; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola | |
| Development of therapeutic agents blocking SOS activation | 1-gen-2019 | Maso, L.; Bellio, P.; Linciano, P.; D' Acunto, M.; Celenza, G.; Tondi, Donatella; Cendron, L. | |
| Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics | 1-gen-2019 | Borsari, Chiara; Dolores Jimenez-Anton, María; Eick, Julia; Bifeld, Eugenia; Jose Torrado, Juan; Isabel Olías-Molero, Ana; Jesús Corral, María; Santarem, Nuno; Baptista, Catarina; Severi, Leda; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Luciani, Rosaria; Tejera Nevado, Paloma; Zander-Dinse, Dorothea; Franco, Caio H.; Ferrari, Stefania; Moraes, Carolina B.; Cordeiro-da-Silva, Anabela; Ponterini, Glauco; Clos, Joachim; María Alunda, Jose; Paola Costi, Maria | |
| Druggability profile of stilbene-derived PPAR agonists: Determination of physicochemical properties and PAMPA study | 1-gen-2019 | Linciano, P.; De Filippis, B.; Ammazzalorso, A.; Amoia, P.; Cilurzo, F.; Fantacuzzi, M.; Giampietro, L.; Maccallini, C.; Petit, C.; Amoroso, R. | |
| Effect of stilbene and chalcone scaffolds incorporation in clofibric acid on PPARα agonistic activity | 1-gen-2014 | Giampietro, Letizia; D'Angelo, Alessandra; Giancristofaro, Antonella; Ammazzalorso, Alessandra; DE FILIPPIS, Barbara; DI MATTEO, Mauro; Fantacuzzi, Marialuigia; Linciano, Pasquale; Maccallini, Cristina; Amoroso, Rosa |