LINCIANO, PASQUALE
LINCIANO, PASQUALE
DIPARTIMENTO DI SCIENZE DEL FARMACO
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity
2019-01-01 Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L.
1,3-Dithiolane as a Privileged Scaffold in Bioactive Derivatives: Chiral Resolution and Assignment of Absolute Configuration
2024-01-01 Listro, R.; Rossino, G.; Cavalloro, V.; Rossi, D.; Boiocchi, M.; Robescu, M. S.; Bavaro, T.; Franchini, S.; Sorbi, C.; De Amici, M.; Linciano, P.; Collina, S.
4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases
2020-01-01 Linciano, Pasquale; Gianquinto, Eleonora; Montanari, Martina; Maso, Lorenzo; Bellio, Pierangelo; Cebrián-Sastre, Esmeralda; Celenza, Giuseppe; Blázquez, Jesús; Cendron, Laura; Spyrakis, Francesca; Tondi, Donatella
A green Heck reaction protocol towards trisubstituted alkenes, versatile pharmaceutical intermediates
2024-01-01 Rossino, G.; Marrubini, G.; Brindisi, M.; Granje, M.; Linciano, P.; Rossi, D.; Collina, S.
A multidisciplinary approach to the design of novel inhibitors for KPC-2
2017-01-01 Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella
A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol
2019-01-01 Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G.
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
2019-01-01 Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz
An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases
2016-01-01 Quotadamo, Antonio; Linciano, Pasquale; Davoli, Paolo; Tondi, Donatella; Costi, Maria Paola; Venturelli, Alberto
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog
2019-01-01 Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G.
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections
2018-01-01 Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola
Biophysical Assays for Investigating Modulators of Macromolecular Complexes: An Overview
2024-01-01 Garbagnoli, Martina; Linciano, Pasquale; Listro, Roberta; Rossino, Giacomo; Vasile, Francesca; Collina, Simona
Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization
2021-01-01 Rossino, G.; Rui, M.; Linciano, P.; Rossi, D.; Boiocchi, M.; Peviani, M.; Poggio, E.; Curti, D.; Schepmann, D.; Wünsch, B.; González-Avendaño, M.; Vergara-Jaque, A.; Caballero, J.; Collina, S.
BS148 Reduces the Aggressiveness of Metastatic Melanoma via Sigma-2 Receptor Targeting
2023-01-01 Sorbi, Claudia; Belluti, Silvia; Atene, Claudio Giacinto; Marocchi, Federica; Linciano, Pasquale; Roy, Neena; Paradiso, Elia; Casarini, Livio; Ronsisvalle, Simone; Zanocco-Marani, Tommaso; Brasili, Livio; Lanfrancone, Luisa; Imbriano, Carol; Di Rocco, Giulia; Franchini, Silvia
Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry
2019-01-01 Citti, C.; Linciano, P.; Panseri, S.; Vezzalini, F.; Forni, F.; Vandelli, M. A.; Cannazza, G.
Chemical and spectroscopic characterization data of ‘cannabidibutol’, a novel cannabidiol butyl analog
2019-01-01 Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G.
Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies
2022-01-01 Linciano, P.; Nasti, R.; Listro, R.; Amadio, M.; Pascale, A.; Potenza, D.; Vasile, F.; Minneci, M.; Ann, J.; Lee, J.; Zhou, X.; Mitchell, G. A.; Blumberg, P. M.; Rossi, D.; Collina, S.
COMPOSTI AD ATTIVITÀ ANTIPARASSITARIA
2019-01-01 Paola Costi, Maria; Costantino, Luca; Linciano, Pasquale; Ferrari, Stefania; Cordeiro da Silva, Anabela
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients?
2023-01-01 D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona
Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth
2019-01-01 Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D’Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Paola Costi, Maria
Design of 2-Aminobenzothiazole Derivatives Targeting Trypanosomatid PTR1 by a Multidisciplinary Fragment Hybridization Approach
2025-01-01 Panecka-Hofman, Joanna; Linciano, Pasquale; Pöhner, Ina; Dyguda-Kazimierowicz, Edyta; Jedwabny, Wiktoria; Landi, Giacomo; Santarem, Nuno; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Luciani, Rosaria; Ferrari, Stefania; Aiello, Daniele; Mangani, Stefano; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Costi, Maria Paola; Wade, Rebecca C.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity | 1-gen-2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L. | |
| 1,3-Dithiolane as a Privileged Scaffold in Bioactive Derivatives: Chiral Resolution and Assignment of Absolute Configuration | 1-gen-2024 | Listro, R.; Rossino, G.; Cavalloro, V.; Rossi, D.; Boiocchi, M.; Robescu, M. S.; Bavaro, T.; Franchini, S.; Sorbi, C.; De Amici, M.; Linciano, P.; Collina, S. | |
| 4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases | 1-gen-2020 | Linciano, Pasquale; Gianquinto, Eleonora; Montanari, Martina; Maso, Lorenzo; Bellio, Pierangelo; Cebrián-Sastre, Esmeralda; Celenza, Giuseppe; Blázquez, Jesús; Cendron, Laura; Spyrakis, Francesca; Tondi, Donatella | |
| A green Heck reaction protocol towards trisubstituted alkenes, versatile pharmaceutical intermediates | 1-gen-2024 | Rossino, G.; Marrubini, G.; Brindisi, M.; Granje, M.; Linciano, P.; Rossi, D.; Collina, S. | |
| A multidisciplinary approach to the design of novel inhibitors for KPC-2 | 1-gen-2017 | Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella | |
| A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol | 1-gen-2019 | Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G. | |
| Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform | 1-gen-2019 | Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz | |
| An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases | 1-gen-2016 | Quotadamo, Antonio; Linciano, Pasquale; Davoli, Paolo; Tondi, Donatella; Costi, Maria Paola; Venturelli, Alberto | |
| Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog | 1-gen-2019 | Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G. | |
| Aryl thiosemicarbazones for the treatment of trypanosomatidic infections | 1-gen-2018 | Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola | |
| Biophysical Assays for Investigating Modulators of Macromolecular Complexes: An Overview | 1-gen-2024 | Garbagnoli, Martina; Linciano, Pasquale; Listro, Roberta; Rossino, Giacomo; Vasile, Francesca; Collina, Simona | |
| Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization | 1-gen-2021 | Rossino, G.; Rui, M.; Linciano, P.; Rossi, D.; Boiocchi, M.; Peviani, M.; Poggio, E.; Curti, D.; Schepmann, D.; Wünsch, B.; González-Avendaño, M.; Vergara-Jaque, A.; Caballero, J.; Collina, S. | |
| BS148 Reduces the Aggressiveness of Metastatic Melanoma via Sigma-2 Receptor Targeting | 1-gen-2023 | Sorbi, Claudia; Belluti, Silvia; Atene, Claudio Giacinto; Marocchi, Federica; Linciano, Pasquale; Roy, Neena; Paradiso, Elia; Casarini, Livio; Ronsisvalle, Simone; Zanocco-Marani, Tommaso; Brasili, Livio; Lanfrancone, Luisa; Imbriano, Carol; Di Rocco, Giulia; Franchini, Silvia | |
| Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry | 1-gen-2019 | Citti, C.; Linciano, P.; Panseri, S.; Vezzalini, F.; Forni, F.; Vandelli, M. A.; Cannazza, G. | |
| Chemical and spectroscopic characterization data of ‘cannabidibutol’, a novel cannabidiol butyl analog | 1-gen-2019 | Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G. | |
| Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies | 1-gen-2022 | Linciano, P.; Nasti, R.; Listro, R.; Amadio, M.; Pascale, A.; Potenza, D.; Vasile, F.; Minneci, M.; Ann, J.; Lee, J.; Zhou, X.; Mitchell, G. A.; Blumberg, P. M.; Rossi, D.; Collina, S. | |
| COMPOSTI AD ATTIVITÀ ANTIPARASSITARIA | 1-gen-2019 | Paola Costi, Maria; Costantino, Luca; Linciano, Pasquale; Ferrari, Stefania; Cordeiro da Silva, Anabela | |
| Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? | 1-gen-2023 | D'Amato, Maura; Campagnoli, Monica; Iadarola, Paolo; Bignami, PAOLA MARGHERITA; Fumagalli, Marco; Chiarelli, LAURENT ROBERT; Stelitano, Giovanni; Meloni, Federica; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero; Vertui, Valentina; Aliberti, Anna; Fossali, Tommaso; Viglio, Simona | |
| Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth | 1-gen-2019 | Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D’Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Paola Costi, Maria | |
| Design of 2-Aminobenzothiazole Derivatives Targeting Trypanosomatid PTR1 by a Multidisciplinary Fragment Hybridization Approach | 1-gen-2025 | Panecka-Hofman, Joanna; Linciano, Pasquale; Pöhner, Ina; Dyguda-Kazimierowicz, Edyta; Jedwabny, Wiktoria; Landi, Giacomo; Santarem, Nuno; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Luciani, Rosaria; Ferrari, Stefania; Aiello, Daniele; Mangani, Stefano; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Costi, Maria Paola; Wade, Rebecca C. |