Sfoglia per Autore
A red-NIR fluorescent dye detecting nuclear DNA G-quadruplexes: in vitro analysis and cell imaging
2017-01-01 Doria, Filippo; Nadai, M.; Zuffo, Michela; Perrone, R.; Freccero, Mauro; Richter, S. N.
Synthesis, Binding Properties, and Differences in Cell Uptake of G-Quadruplex Ligands Based on Carbohydrate Naphthalene Diimide Conjugates
2017-01-01 Arévalo Ruiz, Matilde; Doria, Filippo; Belmonte Reche, Efres; De Rache, Aurore; Campos Salinas, Jenny; Lucas, Ricardo; Falomir, Eva; Carda, Miguel; Pérez Victoria, José María; Mergny, Jean Louis; Freccero, Mauro; Morales, Juan Carlos
A Catalytic and Selective Scissoring Molecular Tool for Quadruplex Nucleic Acids
2018-01-01 Nadai, Matteo; Doria, Filippo; Scalabrin, Matteo; Pirota, Valentina; Grande, Vincenzo; Bergamaschi, Greta; Amendola, Valeria; Winnerdy, Fernaldo Richtia; Phan, Anh Tuân; Richter, Sara N.; Freccero, Mauro
Oxadiazole/pyridine-based ligands: A structural tuning for enhancing G-quadruplex binding
2018-01-01 Doria, Filippo; Pirota, Valentina; Petenzi, Michele; Teulade-Fichou, Marie-Paule; Verga, Daniela; Freccero, Mauro
Controlled Pore Glass-based oligonucleotide affinity support: towards High Throughput Screening methods for the identification of conformation-selective G-quadruplex ligands
2018-01-01 Platella, Chiara; Musumeci, Domenica; Arciello, Angela; Doria, Filippo; Freccero, Mauro; Randazzo, Antonio; Amato, Jussara; Pagano, Bruno; Montesarchio, Daniela
Down-Regulation of the Androgen Receptor by G-Quadruplex Ligands Sensitizes Castration-Resistant Prostate Cancer Cells to Enzalutamide
2018-01-01 Tassinari, Martina; Cimino-Reale, Graziella; Nadai, Matteo; Doria, Filippo; Butovskaya, Elena; Recagni, Marta; Freccero, Mauro; Zaffaroni, Nadia; Richter, Sara N.; Folini, Marco
More is not always better: finding the right trade-off between affinity and selectivity of a G-quadruplex ligand
2018-01-01 Zuffo, Michela; Guédin, Aurore; Leriche, Emma-Dune; Doria, Filippo; Pirota, Valentina; Gabelica, Valérie; Mergny, Jean-Louis; Freccero, Mauro
A Fragment-Based Approach for the Development of G-Quadruplex Ligands: Role of the Amidoxime Moiety
2018-01-01 Tassinari, Martina; Lena, Alberto; Butovskaya, Elena; Pirota, Valentina; Nadai, Matteo; Freccero, Mauro; Doria, Filippo; Richter, Sara N.
G-Quadruplex Identification in the Genome of Protozoan Parasites Points to Naphthalene Diimide Ligands as New Antiparasitic Agents
2018-01-01 Belmonte-Reche, Efres; Martínez-García, Marta; Guédin, Aurore; Zuffo, Michela; Arévalo-Ruiz, Matilde; Doria, Filippo; Campos-Salinas, Jenny; Maynadier, Marjorie; López-Rubio, José Juan; Freccero, Mauro; Mergny, Jean-Louis; Pérez-Victoria, José María; Morales, Juan Carlos
Naphthalene diimide-derivatives G-quadruplex ligands induce cell proliferation inhibition, mild telomeric dysfunction and cell cycle perturbation in U251MG glioma cells
2018-01-01 Muoio, Daniela; Berardinelli, Francesco; Leone, Stefano; Coluzzi, Elisa; di Masi, Alessandra; Doria, Filippo; Freccero, Mauro; Sgura, Antonella; Folini, Marco; Antoccia, Antonio
Photoresponsive molecular devices targeting nucleic acid secondary structures
2019-01-01 Zuffo, M.; Pirota, V.; Doria, F.
The Oncogenic Signaling Pathways in BRAF-Mutant Melanoma Cells are Modulated by Naphthalene Diimide-Like G-Quadruplex Ligands
2019-01-01 Recagni, M.; Tassinari, M.; Doria, F.; Cimino-Reale, G.; Zaffaroni, N.; Freccero, M.; Folini, M.; Richter, S. N.
Naphthalene diimides as multimodal G-quadruplex-selective ligands
2019-01-01 Pirota, V.; Nadai, M.; Doria, F.; Richter, S. N.
Synthesis and photocytotoxic activity of [1,2,3]triazolo[4,5-h][1,6]naphthyridines and [1,3]oxazolo[5,4-h][1,6]naphthyridines
2019-01-01 Frasson, Ilaria; Spanò, Virginia; Di Martino, Simona; Nadai, Matteo; Doria, Filippo; Parrino, Barbara; Carbone, Anna; Cascioferro, Stella Maria; Diana, Patrizia; Cirrincione, Girolamo; Freccero, Mauro; Barraja, Paola; Richter, Sara N.; Montalbano, Alessandra
Dyads of G-Quadruplex Ligands Triggering DNA Damage Response and Tumour Cell Growth Inhibition at Subnanomolar Concentration
2019-01-01 Doria, F.; Salvati, E.; Pompili, L.; Pirota, V.; D'Angelo, C.; Manoli, F.; Nadai, M.; Richter, S. N.; Biroccio, A.; Manet, I.; Freccero, M.
Carbohydrate-naphthalene diimide conjugates as potential antiparasitic drugs: Synthesis, evaluation and structure-activity studies
2019-01-01 Zuffo, M.; Stucchi, A.; Campos-Salinas, J.; Cabello-Donayre, M.; Martínez-García, M.; Belmonte-Reche, E.; Pérez-Victoria, J. M.; Mergny, J. L.; Freccero, M.; Morales, J. C.; Doria, F.
Trifunctionalized Naphthalene Diimides and Dimeric Analogues as G-Quadruplex-Targeting Anticancer Agents Selected by Affinity Chromatography
2020-01-01 Platella, Chiara; Pirota, Valentina; Musumeci, Domenica; Rizzi, Federica; Iachettini, Sara; Zizza, Pasquale; Biroccio, Annamaria; Freccero, Mauro; Montesarchio, Daniela; Doria, Filippo
Triterpenic saponins from Medicago marina L
2020-01-01 Tava, A.; Biazzi, E.; Ronga, D.; Mella, M.; Doria, F.; Accogli, R.; Argentieri, M. P.; Avato, P.
Phytochemical characterization and in vitro antioxidant properties of four Brassica wild species from Italy
2020-01-01 Picchi, V.; Scalzo, R. L.; Tava, A.; Doria, F.; Argento, S.; Toscano, S.; Treccarichi, S.; Branca, F.
Groundbreaking Anticancer Activity of Highly Diversified Oxadiazole Scaffolds
2020-01-01 Benassi, Alessandra; Doria, Filippo; Pirota, Valentina
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A red-NIR fluorescent dye detecting nuclear DNA G-quadruplexes: in vitro analysis and cell imaging | 1-gen-2017 | Doria, Filippo; Nadai, M.; Zuffo, Michela; Perrone, R.; Freccero, Mauro; Richter, S. N. | |
Synthesis, Binding Properties, and Differences in Cell Uptake of G-Quadruplex Ligands Based on Carbohydrate Naphthalene Diimide Conjugates | 1-gen-2017 | Arévalo Ruiz, Matilde; Doria, Filippo; Belmonte Reche, Efres; De Rache, Aurore; Campos Salinas, Jenny; Lucas, Ricardo; Falomir, Eva; Carda, Miguel; Pérez Victoria, José María; Mergny, Jean Louis; Freccero, Mauro; Morales, Juan Carlos | |
A Catalytic and Selective Scissoring Molecular Tool for Quadruplex Nucleic Acids | 1-gen-2018 | Nadai, Matteo; Doria, Filippo; Scalabrin, Matteo; Pirota, Valentina; Grande, Vincenzo; Bergamaschi, Greta; Amendola, Valeria; Winnerdy, Fernaldo Richtia; Phan, Anh Tuân; Richter, Sara N.; Freccero, Mauro | |
Oxadiazole/pyridine-based ligands: A structural tuning for enhancing G-quadruplex binding | 1-gen-2018 | Doria, Filippo; Pirota, Valentina; Petenzi, Michele; Teulade-Fichou, Marie-Paule; Verga, Daniela; Freccero, Mauro | |
Controlled Pore Glass-based oligonucleotide affinity support: towards High Throughput Screening methods for the identification of conformation-selective G-quadruplex ligands | 1-gen-2018 | Platella, Chiara; Musumeci, Domenica; Arciello, Angela; Doria, Filippo; Freccero, Mauro; Randazzo, Antonio; Amato, Jussara; Pagano, Bruno; Montesarchio, Daniela | |
Down-Regulation of the Androgen Receptor by G-Quadruplex Ligands Sensitizes Castration-Resistant Prostate Cancer Cells to Enzalutamide | 1-gen-2018 | Tassinari, Martina; Cimino-Reale, Graziella; Nadai, Matteo; Doria, Filippo; Butovskaya, Elena; Recagni, Marta; Freccero, Mauro; Zaffaroni, Nadia; Richter, Sara N.; Folini, Marco | |
More is not always better: finding the right trade-off between affinity and selectivity of a G-quadruplex ligand | 1-gen-2018 | Zuffo, Michela; Guédin, Aurore; Leriche, Emma-Dune; Doria, Filippo; Pirota, Valentina; Gabelica, Valérie; Mergny, Jean-Louis; Freccero, Mauro | |
A Fragment-Based Approach for the Development of G-Quadruplex Ligands: Role of the Amidoxime Moiety | 1-gen-2018 | Tassinari, Martina; Lena, Alberto; Butovskaya, Elena; Pirota, Valentina; Nadai, Matteo; Freccero, Mauro; Doria, Filippo; Richter, Sara N. | |
G-Quadruplex Identification in the Genome of Protozoan Parasites Points to Naphthalene Diimide Ligands as New Antiparasitic Agents | 1-gen-2018 | Belmonte-Reche, Efres; Martínez-García, Marta; Guédin, Aurore; Zuffo, Michela; Arévalo-Ruiz, Matilde; Doria, Filippo; Campos-Salinas, Jenny; Maynadier, Marjorie; López-Rubio, José Juan; Freccero, Mauro; Mergny, Jean-Louis; Pérez-Victoria, José María; Morales, Juan Carlos | |
Naphthalene diimide-derivatives G-quadruplex ligands induce cell proliferation inhibition, mild telomeric dysfunction and cell cycle perturbation in U251MG glioma cells | 1-gen-2018 | Muoio, Daniela; Berardinelli, Francesco; Leone, Stefano; Coluzzi, Elisa; di Masi, Alessandra; Doria, Filippo; Freccero, Mauro; Sgura, Antonella; Folini, Marco; Antoccia, Antonio | |
Photoresponsive molecular devices targeting nucleic acid secondary structures | 1-gen-2019 | Zuffo, M.; Pirota, V.; Doria, F. | |
The Oncogenic Signaling Pathways in BRAF-Mutant Melanoma Cells are Modulated by Naphthalene Diimide-Like G-Quadruplex Ligands | 1-gen-2019 | Recagni, M.; Tassinari, M.; Doria, F.; Cimino-Reale, G.; Zaffaroni, N.; Freccero, M.; Folini, M.; Richter, S. N. | |
Naphthalene diimides as multimodal G-quadruplex-selective ligands | 1-gen-2019 | Pirota, V.; Nadai, M.; Doria, F.; Richter, S. N. | |
Synthesis and photocytotoxic activity of [1,2,3]triazolo[4,5-h][1,6]naphthyridines and [1,3]oxazolo[5,4-h][1,6]naphthyridines | 1-gen-2019 | Frasson, Ilaria; Spanò, Virginia; Di Martino, Simona; Nadai, Matteo; Doria, Filippo; Parrino, Barbara; Carbone, Anna; Cascioferro, Stella Maria; Diana, Patrizia; Cirrincione, Girolamo; Freccero, Mauro; Barraja, Paola; Richter, Sara N.; Montalbano, Alessandra | |
Dyads of G-Quadruplex Ligands Triggering DNA Damage Response and Tumour Cell Growth Inhibition at Subnanomolar Concentration | 1-gen-2019 | Doria, F.; Salvati, E.; Pompili, L.; Pirota, V.; D'Angelo, C.; Manoli, F.; Nadai, M.; Richter, S. N.; Biroccio, A.; Manet, I.; Freccero, M. | |
Carbohydrate-naphthalene diimide conjugates as potential antiparasitic drugs: Synthesis, evaluation and structure-activity studies | 1-gen-2019 | Zuffo, M.; Stucchi, A.; Campos-Salinas, J.; Cabello-Donayre, M.; Martínez-García, M.; Belmonte-Reche, E.; Pérez-Victoria, J. M.; Mergny, J. L.; Freccero, M.; Morales, J. C.; Doria, F. | |
Trifunctionalized Naphthalene Diimides and Dimeric Analogues as G-Quadruplex-Targeting Anticancer Agents Selected by Affinity Chromatography | 1-gen-2020 | Platella, Chiara; Pirota, Valentina; Musumeci, Domenica; Rizzi, Federica; Iachettini, Sara; Zizza, Pasquale; Biroccio, Annamaria; Freccero, Mauro; Montesarchio, Daniela; Doria, Filippo | |
Triterpenic saponins from Medicago marina L | 1-gen-2020 | Tava, A.; Biazzi, E.; Ronga, D.; Mella, M.; Doria, F.; Accogli, R.; Argentieri, M. P.; Avato, P. | |
Phytochemical characterization and in vitro antioxidant properties of four Brassica wild species from Italy | 1-gen-2020 | Picchi, V.; Scalzo, R. L.; Tava, A.; Doria, F.; Argento, S.; Toscano, S.; Treccarichi, S.; Branca, F. | |
Groundbreaking Anticancer Activity of Highly Diversified Oxadiazole Scaffolds | 1-gen-2020 | Benassi, Alessandra; Doria, Filippo; Pirota, Valentina |
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