IRIS
LINCIANO, PASQUALE
 Distribuzione geografica
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Continente #
NA - Nord America 873
EU - Europa 475
AS - Asia 167
Continente sconosciuto - Info sul continente non disponibili 5
SA - Sud America 3
Totale 1.523
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Nazione #
US - Stati Uniti d'America 872
IE - Irlanda 294
CN - Cina 95
IT - Italia 64
SG - Singapore 59
FI - Finlandia 56
DE - Germania 32
AT - Austria 9
BE - Belgio 9
EU - Europa 5
IN - India 5
FR - Francia 4
CO - Colombia 2
HK - Hong Kong 2
SI - Slovenia 2
TR - Turchia 2
AE - Emirati Arabi Uniti 1
CZ - Repubblica Ceca 1
EC - Ecuador 1
IL - Israele 1
MX - Messico 1
NL - Olanda 1
PH - Filippine 1
SE - Svezia 1
SK - Slovacchia (Repubblica Slovacca) 1
TW - Taiwan 1
UA - Ucraina 1
Totale 1.523
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Città #
Dublin 294
Chandler 257
Ashburn 130
Boardman 82
Shanghai 63
Helsinki 56
Singapore 43
New York 29
Pavia 24
Lawrence 23
Medford 23
Princeton 23
Seattle 21
Wilmington 16
Washington 13
Brussels 9
Munich 9
Vienna 8
Dallas 7
Los Angeles 7
Beijing 6
Bolzaneto 5
Chicago 5
Pune 5
Woodbridge 5
Ann Arbor 3
Milan 3
Norwalk 3
Torino 3
Barranquilla 2
Cernusco sul Naviglio 2
Fairfield 2
Florence 2
Guiyang 2
Houston 2
Istanbul 2
Murska Sobota 2
Paris 2
Piscataway 2
Reggio Emilia 2
Rome 2
Rozzano 2
Santa Clara 2
Siena 2
Turin 2
West Jordan 2
Andover 1
Atlanta 1
Ballabio 1
Berlin 1
Bologna 1
Bratislava 1
Braunschweig 1
Brno 1
Chengdu 1
Citta 1
Dubai 1
Englewood 1
Falkenstein 1
Fuzhou 1
Gunzenhausen 1
Jacksonville 1
Luoyang 1
Mexico City 1
Nanchang 1
Omaha 1
Padova 1
Palermo 1
Phoenix 1
Quito 1
Redmond 1
Shenyang 1
Stockholm 1
Taipei 1
Ugong Norte 1
Varese 1
Totale 1.239
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Nome #
Identification of N,N-arylalkyl-picolinamide derivatives targeting the RNA-binding protein HuR, by combining biophysical fragment-screening and molecular hybridization 49
Effects of Bisphenols on RACK1 Expression and Their Immunological Implications in THP-1 Cells 48
Identification of a Potent and Selective 5-HT1AReceptor Agonist with in Vitro and in Vivo Antinociceptive Activity 44
4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases 42
Microwave-Assisted Extraction and HPLC-UV-CD Determination of (S)-usnic Acid in Cladonia foliacea 41
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity 39
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign 38
Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents 38
Chiral 2-phenyl-3-hydroxypropyl esters as PKC-alpha modulators: HPLC enantioseparation, NMR absolute configuration assignment, and molecular docking studies 38
Tackling Antimicrobial Resistance with Small Molecules Targeting LsrK: Challenges and Opportunities 37
Investigation of the effect of different linker chemotypes on the inhibition of Histone Deacetylases (HDACs) 37
Evidence of pyrimethamine and cycloguanil analogues as dual inhibitors of trypanosoma brucei pteridine reductase and dihydrofolate reductase 37
Sigma-1 receptor antagonists: promising players in fighting neuropathic pain 36
Sigma-1 receptor agonists acting on aquaporin-mediated h2o2 permeability: New tools for counteracting oxidative stress 36
COMPOSTI AD ATTIVITÀ ANTIPARASSITARIA 35
Druggability profile of stilbene-derived PPAR agonists: Determination of physicochemical properties and PAMPA study 33
The novel heptyl phorolic acid cannabinoids content in different Cannabis sativa L. accessions 33
An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases 32
Setup and Validation of a Reliable Docking Protocol for the Development of Neuroprotective Agents by Targeting the Sigma-1 Receptor (S1R) 31
Bitopic Sigma 1 Receptor Modulators to Shed Light on Molecular Mechanisms Underpinning Ligand Binding and Receptor Oligomerization 31
Effect of the rigidification of propranolol, a mixed β-adrenoceptor and 5-HT1AR antagonist 30
EFFECTS OF ENDOCRINE ACTIVE CONTAMINATING PESTICIDES ON RACK1 EXPRESSION AND IMMUNOLOGICAL CONSEQUENCES IN THP-1 CELLS 30
Cannabinoid profiling of hemp seed oil by liquid chromatography coupled to high-resolution mass spectrometry 30
Scouting Sigma Receptor Ligands As New Tools For The Treatment Of Neurodegenerative Diseases And Cancer 29
Could the Oxidation of α1-Antitrypsin Prevent the Binding of Human Neutrophil Elastase in COVID-19 Patients? 29
High-resolution crystal structure of Trypanosoma brucei pteridine reductase 1 in complex with an innovative tricyclic-based inhibitor 28
Chemical and spectroscopic characterization data of ‘cannabidibutol’, a novel cannabidiol butyl analog 27
Origin of Δ9-Tetrahydrocannabinol Impurity in Synthetic Cannabidiol 27
Ten Years with New Delhi Metallo-β-lactamase-1 (NDM-1): From Structural Insights to Inhibitor Design 27
Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth 26
A multidisciplinary approach to the design of novel inhibitors for KPC-2 25
New weapons against antimicrobial resistance: 
Targeting SOS response to recover b
 actericidal activity of antibiotics
 24
Is cannabidiol a scheduled controlled substance? Origin makes the difference 24
Development of therapeutic agents blocking SOS activation 23
Identification of a new cannabidiol n-hexyl homolog in a medicinal cannabis variety with an antinociceptive activity in mice: cannabidihexol 23
Effect of stilbene and chalcone scaffolds incorporation in clofibric acid on PPARα agonistic activity 22
Geometric Isomerism of an Acetamidino Derivative Determined by NMR Investigations 22
Structural Insights into the Ligand-LsrK Kinase Binding Mode: A Step Forward in the Discovery of Novel Antimicrobial Agents 21
A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol 21
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform 19
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics 17
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections 16
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog 16
From Nature to Synthetic Compounds: Novel 1(N),2,3 Trisubstituted-5-oxopyrrolidines Targeting Multiple Myeloma Cells 14
Sigma receptor and aquaporin modulators: chiral resolution, configurational assignment, and preliminary biological profile of RC752 enantiomers 12
Repurposing the Antiplatelet Agent Ticlopidine to Counteract the Acute Phase of ER Stress Condition: An Opportunity for Fighting Coronavirus Infections and Cancer 12
Novel S1R agonists counteracting NMDA excitotoxicity and oxidative stress: A step forward in the discovery of neuroprotective agents 11
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth 11
Discovery of RC-752, a Novel Sigma-1 Receptor Antagonist with Antinociceptive Activity: A Promising Tool for Fighting Neuropathic Pain 11
Synthesis and structure-activity relationships of fibrate-based analogues inside PPARs 10
Structural development studies of PPARs ligands based on tyrosine scaffold 9
Short- and Long-Term Regulation of HuD: A Molecular Switch Mediated by Folic Acid? 9
Identification of a novel extracellular inhibitor of FGF2/FGFR signaling axis by combined virtual screening and NMR spectroscopy approach 9
Evolving Challenges and Opportunities in Plant-based Drug Discovery and Development 9
Neurodegeneration: can metabolites from Eremurus persicus help? 8
Hits and Lead Discovery in the Identification of New Drugs against the Trypanosomatidic Infections 8
First virtual screening and experimental validation of inhibitors targeting GES-5 carbapenemase 8
Urea-based anticancer agents. Exploring 100-years of research with an eye to the future 8
Excited-state intramolecular proton transfer in a bioactive flavonoid provides fluorescence observables for recognizing its engagement with target proteins 8
Phenyl boronic acids development led to validated leads active in clinical strains overexpressing KPC-2: a step against bacterial resistance 8
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds 8
Sigma receptor and aquaporin modulators: chiral resolution, configurational assignment, and preliminary biological profile of RC752 enantiomers 7
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors 7
Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections 7
Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To InhibitTrypanosoma bruceiPteridine Reductase in Support of Early-Stage Drug Discovery 7
Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARa 7
Peptides as Therapeutic Agents: Challenges and Opportunities in the Green Transition Era 7
Isolation of a High-Affinity Cannabinoid for the Human CB1 Receptor from a Medicinal Cannabis sativa Variety: Δ9-Tetrahydrocannabutol, the Butyl Homologue of Δ9-Tetrahydrocannabinol 6
Biophysical Assays for Investigating Modulators of Macromolecular Complexes: An Overview 6
Phenylboronic Acids Probing Molecular Recognition against Class A and Class C beta-Lactamases 6
In silico identification and experimental validation of hits active against KPC-2 β-lactamase 6
Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1 5
The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents 5
Use of primary amines for the selective N-Alkylation of anilines by a reusable heterogeneous catalyst 5
Optimization of N-alkylation in the Synthesis of Methotrexate and Pteridine-based Derivatives Under Microwave-Irradiation 5
Identification of HuR-RNA Interfering Compounds by Dynamic Combinatorial Chemistry and Fluorescence Polarization 4
Totale 1.574
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Categoria #
all - tutte 11.856
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 11.856
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/202132 0 0 0 17 3 0 4 4 4 0 0 0
2021/2022120 0 0 16 0 1 3 1 13 2 4 22 58
2022/2023729 33 45 14 65 56 76 0 47 341 9 27 16
2023/2024506 23 92 21 27 34 124 63 40 6 21 22 33
2024/2025187 23 93 20 24 27 0 0 0 0 0 0 0
Totale 1.574